Compile Data Set for Download or QSAR
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Found 24 Enz. Inhib. hit(s) with all data for entry = 50046663
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124215(CHEMBL3622866)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124350(CHEMBL3622839)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50330063(1-(4-(Aminomethyl)benzyl)-2-butyl-1H-imidazo[4,5-c...)
Affinity DataEC50:  55nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124216(CHEMBL3622865)
Affinity DataEC50:  621nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124217(CHEMBL3622863)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124218(CHEMBL3622862)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124219(CHEMBL3622861)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124220(CHEMBL3622860)
Affinity DataEC50:  1.02E+3nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124221(CHEMBL3622859)
Affinity DataEC50:  519nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124222(CHEMBL3622858)
Affinity DataEC50:  727nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124223(CHEMBL3622857)
Affinity DataEC50:  2.86E+3nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124224(CHEMBL3622856)
Affinity DataEC50:  2.18E+3nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124225(CHEMBL3622855)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124340(CHEMBL3622854)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124341(CHEMBL3622853)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124342(CHEMBL3622852)
Affinity DataEC50:  91nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124343(CHEMBL3622851)
Affinity DataEC50:  699nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124344(CHEMBL3622847)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124345(CHEMBL3622846)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124346(CHEMBL3622844)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124347(CHEMBL3622842)
Affinity DataEC50:  250nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124348(CHEMBL3622841)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50124349(CHEMBL3622840)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50330062(1-(3-(Aminomethyl)benzyl)-2-butyl-1H-imidazo[4,5-c...)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human TLR8 transfected in HEK293 cells assessed as activation of NF-kB by reporter gene assayMore data for this Ligand-Target Pair