Compile Data Set for Download or QSAR
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Found 24 Enz. Inhib. hit(s) with all data for entry = 50046782
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130903(CHEMBL3632950)
Affinity DataKi:  1.76E+3nMAssay Description:Fixed inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by Dixon and Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130903(CHEMBL3632950)
Affinity DataIC50:  2.02E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130915(CHEBI:3122 | CHEMBL1231178)
Affinity DataIC50:  4.03E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130901(CHEMBL3632948)
Affinity DataIC50:  4.58E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130908(CHEMBL3632954)
Affinity DataIC50:  4.63E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130884(CHEMBL3632946)
Affinity DataIC50:  4.72E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130919(CHEMBL3632942)
Affinity DataIC50:  8.68E+3nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130922(CHEMBL3632941)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130905(CHEMBL3632952)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130913(CHEMBL3632958)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130911(CHEMBL3632956)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130894(CHEMBL3632627)
Affinity DataIC50:  1.74E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130914(CHEMBL3632959)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130906(CHEMBL3632953)
Affinity DataIC50:  2.27E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130912(CHEMBL3632957)
Affinity DataIC50:  2.43E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130900(CHEMBL3632947)
Affinity DataIC50:  2.57E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130918(CHEMBL3632943)
Affinity DataIC50:  3.34E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130909(CHEMBL2074634)
Affinity DataIC50:  3.62E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130910(CHEMBL3632955)
Affinity DataIC50:  4.11E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130902(CHEMBL3632949)
Affinity DataIC50:  5.88E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130904(CHEMBL3632951)
Affinity DataIC50:  7.16E+4nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130916(CHEMBL3632945)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130907(ALISOL A)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
Liaoning University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50130917(CHEMBL3632944)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of human carboxylesterase 2 using 4-benzoyl-N-butyl-1,8-naphthalimide as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed