Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50006414
TargetZinc metalloproteinase dpy-31(Brugia malayi)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50216823(2-(5-{(1R)-4-cyclohexyl-1-[2-(hydroxyamino)-2-oxoe...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499818(CHEMBL3740110)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Brugia malayi)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499820(CHEMBL3740431)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499820(CHEMBL3740431)
Affinity DataIC50:  3.16E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50216823(2-(5-{(1R)-4-cyclohexyl-1-[2-(hydroxyamino)-2-oxoe...)
Affinity DataIC50:  3.98E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Brugia malayi)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499818(CHEMBL3740110)
Affinity DataIC50:  7.94E+4nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50063917((2S,3R)-N(4)-[(2S)-3,3-dimethyl-1-(methylamino)-1-...)
Affinity DataIC50:  7.94E+4nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Brugia malayi)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50063917((2S,3R)-N(4)-[(2S)-3,3-dimethyl-1-(methylamino)-1-...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Brugia malayi)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499819(CHEMBL3740244)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetZinc metalloproteinase dpy-31(Teladorsagia circumcincta)
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50499819(CHEMBL3740244)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of recombinant Teladorsagia circumcincta DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preinc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed