TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 9.90nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 109nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 122nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 201nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 207nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 212nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 222nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 342nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 424nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair