Found 8 Enz. Inhib. hit(s) with all data for entry = 50010062 
Affinity DataIC50: 3.80nMAssay Description:Activity at biotinylated 6His-tagged human RORgamma LBD (259 to 518 residues) assessed as induction of biotinylated SRC1 peptide recruitment incubate...More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 7nMAssay Description:Activity at biotinylated APC-labeled human RORgamma LBD assessed as of Induction of biotinylated SRC1 peptide recruitment incubated for 1 hr by TR-FR...More data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Activity at RORgamma in human PBMC assessed as induction of IL17A production after 4 days by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inverse agonist activity at GAL4-fused human RORgamma expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 18hr...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Activity at APC-labeled 6His-tagged human RORgamma LBD (263 to 518 residues) expressed in Escherichia coli BL21 (DE3) cells assessed as induction of ...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Displacement of [3H]T0901317 from N-6HN-MBP-Avi-TCS-tagged human RORgamma LBD (P260 to K518 residues) preincubated for 30 mins followed by ligand add...More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) expressed in human Jurkat cells assessed as inhibition of IL-17F production after 20 hrs by luc...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Activity at 6His-tagged human RORgamma LBD (262 to 507 residues) expressed in Escherichia coli BL21 (DE3) cells assessed as induction of biotinylated...More data for this Ligand-Target Pair
