Found 56 Enz. Inhib. hit(s) with all data for entry = 50047929 
Affinity DataIC50: 3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 123nMAssay Description:Inhibition of activated TAFI in human blood by clot lysis assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Sanofi R & D
Curated by ChEMBL
Sanofi R & D
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human ERG expressed in CHO cells by patch clamp methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate assessed as suppression of 1'-hydroxymidazolam formation after 10 mins by...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins in presence of 1% human serum albumin by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of activated human plasma TAFI incubated for 15 mins by chromogenic assayMore data for this Ligand-Target Pair
