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Found 8 Enz. Inhib. hit(s) with all data for entry = 50048001
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50200519(CHEMBL3915703)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of p110delta (unknown origin) assessed as decrease in ATP consumption after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50200518(CHEMBL3945937)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of p110delta (unknown origin) assessed as decrease in ATP consumption after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50200518(CHEMBL3945937)
Affinity DataIC50:  4.38E+4nMAssay Description:Inhibition of p110alpha (unknown origin) assessed as decrease in ATP consumption after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50200519(CHEMBL3915703)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of p110beta (unknown origin) assessed as decrease in ATP consumption after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50200519(CHEMBL3915703)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of p110gamma (unknown origin) assessed as decrease in ATP consumption after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50200519(CHEMBL3915703)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of p110alpha (unknown origin) assessed as decrease in ATP consumption after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50200518(CHEMBL3945937)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of p110gamma (unknown origin) assessed as decrease in ATP consumption after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50200518(CHEMBL3945937)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of p110beta (unknown origin) assessed as decrease in ATP consumption after 60 mins by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed