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Found 8 Enz. Inhib. hit(s) with all data for entry = 50048196
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of human recombinant full-length N-terminal His-tagged BTK expressed in baculovirus infected Sf9 insect cells measured after 60 mins by AD...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50161162(AVL-292 | CC-292 | Spebrutinib | US10596172, Compo...)
Affinity DataIC50:  0.720nMAssay Description:Inhibition of human recombinant full-length N-terminal His-tagged BTK expressed in baculovirus infected Sf9 insect cells measured after 60 mins by AD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50207562(CHEMBL3904000)
Affinity DataIC50:  0.820nMAssay Description:Inhibition of human recombinant full-length N-terminal His-tagged BTK expressed in baculovirus infected Sf9 insect cells measured after 60 mins by AD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50207563(CHEMBL3932000)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human recombinant full-length N-terminal His-tagged BTK expressed in baculovirus infected Sf9 insect cells measured after 60 mins by AD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50207564(CHEMBL3895072)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant full-length N-terminal His-tagged BTK expressed in baculovirus infected Sf9 insect cells measured after 60 mins by AD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50207558(CHEMBL3972321)
Affinity DataIC50:  22nMAssay Description:Inhibition of human recombinant full-length N-terminal His-tagged BTK expressed in baculovirus infected Sf9 insect cells measured after 60 mins by AD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50207566(CHEMBL3895794)
Affinity DataIC50:  32nMAssay Description:Inhibition of human recombinant full-length N-terminal His-tagged BTK expressed in baculovirus infected Sf9 insect cells measured after 60 mins by AD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50207565(CHEMBL3905062)
Affinity DataIC50:  112nMAssay Description:Inhibition of human recombinant full-length N-terminal His-tagged BTK expressed in baculovirus infected Sf9 insect cells measured after 60 mins by AD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed