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Found 68 Enz. Inhib. hit(s) with all data for entry = 50035731
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000091((6S,11R)-3-Cyclopropylmethyl-6-ethyl-8-hydroxy-11-...)
Affinity DataKi:  0.570nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000091((6S,11R)-3-Cyclopropylmethyl-6-ethyl-8-hydroxy-11-...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018786(CHEMBL538309 | N-(2-Azocan-1-yl-cyclohexyl)-N-meth...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018768(CHEMBL556957 | N-(2-Azepan-1-yl-cyclohexyl)-2-(4-c...)
Affinity DataKi:  4nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018762(2-Benzofuran-4-yl-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018767(CHEMBL535581 | N-(2-Azocan-1-yl-cyclohexyl)-N-meth...)
Affinity DataKi:  5.60nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018771(CHEMBL535801 | N-(2-Azepan-1-yl-cyclohexyl)-N-meth...)
Affinity DataKi:  6.40nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)
Affinity DataKi:  7.30nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50008854(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  9.60nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50008854(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  9.60nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 15 min of incubation at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  10nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018762(2-Benzofuran-4-yl-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi:  12nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 60 min of incubation at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018762(2-Benzofuran-4-yl-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi:  12nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018781(CHEMBL557426 | N-Methyl-N-(2-pyrrolidin-1-yl-cyclo...)
Affinity DataKi:  12nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM83436(2-(3,4-dichlorophenyl)-N-methyl-N-[(5R,7S,8S)-7-(1...)
Affinity DataKi:  17nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018778(2-Benzo[b]thiophen-4-yl-N-methyl-N-[2-(methyl-phen...)
Affinity DataKi:  26nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018784(CHEMBL559217 | N-(2-Azepan-1-yl-cyclohexyl)-2-benz...)
Affinity DataKi:  29nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018778(2-Benzo[b]thiophen-4-yl-N-methyl-N-[2-(methyl-phen...)
Affinity DataKi:  30nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018764(2-(3,4-Dichloro-phenoxy)-N-methyl-N-(2-pyrrolidin-...)
Affinity DataKi:  35nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018788(CHEMBL537169 | N-(2-Azepan-1-yl-cyclohexyl)-2-benz...)
Affinity DataKi:  40nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM21130(N-methyl-2-phenyl-N-[(5R,7S,8S)-7-(pyrrolidin-1-yl...)
Affinity DataKi:  52nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018783(CHEMBL539582 | N-[2-(Allyl-methyl-amino)-cyclohexy...)
Affinity DataKi:  52nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018776(CHEMBL537615 | N-(2-Azepan-1-yl-cyclohexyl)-2-(3,5...)
Affinity DataKi:  72nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018763(2-(1H-Indol-3-yl)-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi:  74nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018779(2-Benzo[b]thiophen-4-yl-N-methyl-N-{2-[methyl-(2-t...)
Affinity DataKi:  81nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018779(2-Benzo[b]thiophen-4-yl-N-methyl-N-{2-[methyl-(2-t...)
Affinity DataKi:  82nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  86nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018781(CHEMBL557426 | N-Methyl-N-(2-pyrrolidin-1-yl-cyclo...)
Affinity DataKi:  140nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018772(CHEMBL535130 | N-Methyl-2-(4-nitro-3-trifluorometh...)
Affinity DataKi:  150nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018766(2-Benzo[b]thiophen-4-yl-N-[2-(cyclopropylmethyl-me...)
Affinity DataKi:  190nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018766(2-Benzo[b]thiophen-4-yl-N-[2-(cyclopropylmethyl-me...)
Affinity DataKi:  200nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018783(CHEMBL539582 | N-[2-(Allyl-methyl-amino)-cyclohexy...)
Affinity DataKi:  210nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018780(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-piperidin-1-...)
Affinity DataKi:  250nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018774(2-(4-Chloro-phenoxy)-N-methyl-N-(2-pyrrolidin-1-yl...)
Affinity DataKi:  300nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018785(2-Benzo[b]thiophen-4-yl-N-(2-diethylamino-cyclohex...)
Affinity DataKi:  350nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018777(CHEMBL556802 | N-Methyl-2-phenoxy-N-(2-pyrrolidin-...)
Affinity DataKi:  360nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018768(CHEMBL556957 | N-(2-Azepan-1-yl-cyclohexyl)-2-(4-c...)
Affinity DataKi:  460nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018764(2-(3,4-Dichloro-phenoxy)-N-methyl-N-(2-pyrrolidin-...)
Affinity DataKi:  620nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018771(CHEMBL535801 | N-(2-Azepan-1-yl-cyclohexyl)-N-meth...)
Affinity DataKi:  720nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018773(CHEMBL535133 | N-Methyl-N-(2-pyrrolidin-1-yl-cyclo...)
Affinity DataKi:  720nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018788(CHEMBL537169 | N-(2-Azepan-1-yl-cyclohexyl)-2-benz...)
Affinity DataKi:  810nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018786(CHEMBL538309 | N-(2-Azocan-1-yl-cyclohexyl)-N-meth...)
Affinity DataKi:  880nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50008854(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  880nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  880nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018775(3-(1H-Indol-3-yl)-N-methyl-N-(2-pyrrolidin-1-yl-cy...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50008854(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  1.00E+3nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018772(CHEMBL535130 | N-Methyl-2-(4-nitro-3-trifluorometh...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50018777(CHEMBL556802 | N-Methyl-2-phenoxy-N-(2-pyrrolidin-...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Parke-Davis Research Unit

Curated by ChEMBL
LigandPNGBDBM50008854(2-Benzo[b]thiophen-4-yl-N-methyl-N-(2-pyrrolidin-1...)
Affinity DataKi:  1.00E+3nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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