TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 0.570nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 9.60nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 9.60nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 15 min of incubation at pH 7.2More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 60 min of incubation at pH 7.2More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 72nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 74nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 360nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 720nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: 720nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 810nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 880nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 880nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 880nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Parke-Davis Research Unit
Curated by ChEMBL
Parke-Davis Research Unit
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for the Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 0 min of incubation at pH 7.2More data for this Ligand-Target Pair