Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50001024
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267897(CHEMBL4092297)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267911(CHEMBL4096245)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267896(CHEMBL4064614)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267893(CHEMBL4086083)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267909(CHEMBL4094766)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267895(CHEMBL4084562)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267916(CHEMBL531227 | TCMDC-125004)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267913(CHEMBL602783 | GNF-Pf-3043)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267901(CHEMBL4087066)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267917(CHEMBL4080499)
Affinity DataIC50:  2.11E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267915(CHEMBL4088361)
Affinity DataIC50:  2.82E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267921(CHEMBL4095711)
Affinity DataIC50:  3.56E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267910(CHEMBL4074261)
Affinity DataIC50:  3.69E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267914(CHEMBL4067097)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267912(CHEMBL4069800)
Affinity DataIC50:  5.35E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rattus norvegicus)
Tokyo Medical And Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267894(CHEMBL4102505)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed