Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50001091
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50269302(CHEMBL4060515)
Affinity DataIC50:  276nMAssay Description:Inhibition of human mPGES-1 expressed in 293-F cells using PGH2 as substrate preincubated for 15 mins followed by substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50269300(CHEMBL4077049)
Affinity DataIC50:  284nMAssay Description:Inhibition of human mPGES-1 expressed in 293-F cells using PGH2 as substrate preincubated for 15 mins followed by substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50269301(CIBA-1906 | Thiambutosine)
Affinity DataIC50:  370nMAssay Description:Inhibition of human mPGES-1 expressed in 293-F cells using PGH2 as substrate preincubated for 15 mins followed by substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50269299(CHEMBL4077072)
Affinity DataIC50:  439nMAssay Description:Inhibition of human mPGES-1 expressed in 293-F cells using PGH2 as substrate preincubated for 15 mins followed by substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50269303(CHEMBL4071915)
Affinity DataIC50:  664nMAssay Description:Inhibition of human mPGES-1 expressed in 293-F cells using PGH2 as substrate preincubated for 15 mins followed by substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50269304(CHEMBL4093446)
Affinity DataIC50:  889nMAssay Description:Inhibition of human mPGES-1 expressed in 293-F cells using PGH2 as substrate preincubated for 15 mins followed by substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50269305(CHEMBL1970663)
Affinity DataIC50:  917nMAssay Description:Inhibition of human mPGES-1 expressed in 293-F cells using PGH2 as substrate preincubated for 15 mins followed by substrate addition measured after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed