Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50035605
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50252861(CHEMBL507214 | H-D-Phe-c[Cys-Tyr-DTrp-Orn-Thr-Pen]...)
Affinity DataIC50:  2.80nMAssay Description:Compound was evaluated for the inhibition of binding of [3H]naloxone toOpioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019567(CHEMBL413950 | D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of binding of [3H]-naloxone to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019572(CHEMBL437283 | D-Phe-Cys-Tyr-D-Trp-Lys-Thr-Pen-Thr...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of binding of [3H]-naloxone to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367297(CHEMBL1790572)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of binding of [3H]-naloxone to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataIC50:  6nMAssay Description:Inhibition of binding of [3H]-naloxone to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019575(19-(2-Amino-3-phenyl-propionylamino)-10-butyl-16-(...)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of binding of [3H]-naloxone to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019573(CHEMBL384284 | D-PhGly-Cys-Tyr-D-Trp-Lys-Thr-Pen-T...)
Affinity DataIC50:  350nMAssay Description:Inhibition of binding of [3H]-naloxone to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019570(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataIC50:  539nMAssay Description:Inhibition of binding of [3H]-naloxone to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019569(CHEMBL274400 | D-Phe-Cys-Tyr--Trp-Lys-Thr-Pen-Thr-...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of binding of [3H]-naloxone to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367297(CHEMBL1790572)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019566(2-{[10-(4-Amino-butyl)-19-(2-amino-2-phenyl-acetyl...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of binding of [3H]-naloxone to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019573(CHEMBL384284 | D-PhGly-Cys-Tyr-D-Trp-Lys-Thr-Pen-T...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019567(CHEMBL413950 | D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019575(19-(2-Amino-3-phenyl-propionylamino)-10-butyl-16-(...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019572(CHEMBL437283 | D-Phe-Cys-Tyr-D-Trp-Lys-Thr-Pen-Thr...)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019576(2-{[10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-ph...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of binding of [3H]-naloxone to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50252861(CHEMBL507214 | H-D-Phe-c[Cys-Tyr-DTrp-Orn-Thr-Pen]...)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019576(2-{[10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-ph...)
Affinity DataIC50:  2.75E+4nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019566(2-{[10-(4-Amino-butyl)-19-(2-amino-2-phenyl-acetyl...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019570(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataIC50:  5.80E+4nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50019569(CHEMBL274400 | D-Phe-Cys-Tyr--Trp-Lys-Thr-Pen-Thr-...)
Affinity DataIC50: >7.00E+4nMAssay Description:Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed