Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of EphA2 autophosphorylation at Ser897 in human C13 cells after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
Affinity DataKd: 741nMAssay Description:Binding affinity to NFKBIA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 81nMAssay Description:Binding affinity to recombinant human GST-tagged EphA2 cytoplasmic domain (560 to 976 residues) expressed in baculovirus expression system by fluores...More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
University Of South Florida
Curated by ChEMBL
University Of South Florida
Curated by ChEMBL
Affinity DataKd: 3.62E+3nMAssay Description:Binding affinity to AKT1 (unknown origin)More data for this Ligand-Target Pair