Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50000179
TargetEphrin type-A receptor 2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50246758(CHEMBL4093682)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of EphA2 autophosphorylation at Ser897 in human C13 cells after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50246750(CHEMBL4071045)
Affinity DataKd:  741nMAssay Description:Binding affinity to NFKBIA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-A receptor 2(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50246750(CHEMBL4071045)
Affinity DataKd:  81nMAssay Description:Binding affinity to recombinant human GST-tagged EphA2 cytoplasmic domain (560 to 976 residues) expressed in baculovirus expression system by fluores...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50246750(CHEMBL4071045)
Affinity DataKd:  3.62E+3nMAssay Description:Binding affinity to AKT1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed