Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50002150
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50024330(3-(3-Benzyl-ureido)-3-{2-[2-tert-butoxycarbonylami...)
Affinity DataIC50:  500nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020575(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  750nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020560(4-Benzylcarbamoyl-3-{2-[2-tert-butoxycarbonylamino...)
Affinity DataIC50:  1.00E+3nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020564(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  1.50E+3nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020561(3-{3-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  2.00E+3nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020569(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  2.00E+3nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020573(3-{3-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  5.00E+3nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020574(CHEMBL356844 | N-Benzyl-3-{3-[2-tert-butoxycarbony...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020572(3-{3-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  1.00E+4nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020566(3-{3-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  1.00E+4nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020567(CHEMBL355927 | N-Benzyl-3-{3-[2-tert-butoxycarbony...)
Affinity DataIC50: >1.00E+4nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020571(4-Benzylcarbamoyl-3-{2-[2-tert-butoxycarbonylamino...)
Affinity DataIC50:  1.50E+4nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020563(CHEMBL151619 | N-Benzyl-3-{3-[2-tert-butoxycarbony...)
Affinity DataIC50:  2.00E+4nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020562(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  2.50E+4nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled gCholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020576(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  3.00E+4nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020570(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  5.00E+4nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020577(3-{3-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  5.00E+4nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)

Curated by ChEMBL
LigandPNGBDBM50020568(3-{3-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  1.00E+5nMAssay Description:Invitro inhibition of binding of [125I]-(Nle)-HG-13 labeled Cholecystokinin type B receptor on isolated gastric mucosal cells of rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed