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Found 39 Enz. Inhib. hit(s) with all data for entry = 50000338
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  390nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  2.80E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2B expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  4.70E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  5.90E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2C expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  1.00E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2B expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246919(CHEMBL4099104)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246919(CHEMBL4099104)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2D(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  2.10E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2D expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  2.40E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2C expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2D(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  4.10E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2D expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246917(CHEMBL4068651)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246918(CHEMBL4091369)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246918(CHEMBL4091369)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246914(CHEMBL4088958)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246911(CHEMBL4076785)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246915(CHEMBL4060745)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246918(CHEMBL4091369)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246911(CHEMBL4076785)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246919(CHEMBL4099104)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246916(CHEMBL4102488)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246917(CHEMBL4068651)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246911(CHEMBL4076785)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246914(CHEMBL4088958)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246916(CHEMBL4102488)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246916(CHEMBL4102488)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246914(CHEMBL4088958)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246917(CHEMBL4068651)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  1.31E+5nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  1.54E+5nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246913(CHEMBL4083586)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK3a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintillation c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246913(CHEMBL4083586)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246915(CHEMBL4060745)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-SYM2081 from recombinant homomeric rat GluK1 (Q)1b receptor expressed in baculovirus infected Sf9 insect cell membranes by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246915(CHEMBL4060745)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246913(CHEMBL4083586)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-KA from recombinant homomeric rat GluK2 (V,C,R)a receptor expressed in baculovirus infected Sf9 insect cell membranes by scintil...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataIC50:  1.50E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataIC50:  2.90E+4nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2B expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataIC50:  1.10E+5nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2C expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2D(RAT)
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataIC50:  1.70E+5nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2D expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed