Compile Data Set for Download or QSAR
maximum 50k data
Found 54 Enz. Inhib. hit(s) with all data for entry = 50002739
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462277(CHEMBL4238084)
Affinity DataEC50:  12nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462304(CHEMBL4237902)
Affinity DataEC50:  3.60nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462279(CHEMBL4249199)
Affinity DataEC50:  2.60nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462280(CHEMBL4244929)
Affinity DataEC50:  1.59E+4nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462277(CHEMBL4238084)
Affinity DataEC50:  889nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462281(CHEMBL4245391)
Affinity DataEC50:  15nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462282(CHEMBL4249564)
Affinity DataEC50:  0.512nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462283(CHEMBL4242824)
Affinity DataEC50:  10nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462282(CHEMBL4249564)
Affinity DataEC50:  52nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462282(CHEMBL4249564)
Affinity DataEC50:  2.90nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462284(CHEMBL4248727)
Affinity DataEC50:  55nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462285(CHEMBL4241176)
Affinity DataEC50:  3.40nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462286(CHEMBL4248369)
Affinity DataEC50:  1nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462287(CHEMBL4238856)
Affinity DataEC50:  4.60nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462288(CHEMBL4244608)
Affinity DataEC50:  1.80nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462289(CHEMBL4245968)
Affinity DataEC50:  281nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462285(CHEMBL4241176)
Affinity DataEC50:  8.43E+3nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462290(CHEMBL4250942)
Affinity DataEC50:  8.40nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462291(CHEMBL4248093)
Affinity DataEC50:  299nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462284(CHEMBL4248727)
Affinity DataEC50:  426nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462285(CHEMBL4241176)
Affinity DataEC50:  224nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462291(CHEMBL4248093)
Affinity DataEC50:  11nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462289(CHEMBL4245968)
Affinity DataEC50:  8.70nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462292(CHEMBL4246134)
Affinity DataEC50:  7.80nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462280(CHEMBL4244929)
Affinity DataEC50:  4.60nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462293(CHEMBL4237802)
Affinity DataEC50:  4.70nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462294(CHEMBL4237453)
Affinity DataEC50:  1.40nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462295(CHEMBL4251063)
Affinity DataEC50:  2.90nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462296(CHEMBL4244123)
Affinity DataEC50:  2.20nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462297(CHEMBL4247910)
Affinity DataEC50:  2.90nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462298(CHEMBL4249769)
Affinity DataEC50:  2.5nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462299(CHEMBL4240360)
Affinity DataEC50:  1.5nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462300(CHEMBL4250902)
Affinity DataEC50:  1.40nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462301(CHEMBL4246625)
Affinity DataEC50:  2.10nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462277(CHEMBL4238084)
Affinity DataEC50:  2.35E+4nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462291(CHEMBL4248093)
Affinity DataEC50:  954nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462284(CHEMBL4248727)
Affinity DataEC50:  1.42E+3nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462292(CHEMBL4246134)
Affinity DataEC50:  6.06E+3nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462293(CHEMBL4237802)
Affinity DataEC50:  9.84E+3nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462294(CHEMBL4237453)
Affinity DataEC50:  118nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462278(CHEMBL4241613)
Affinity DataEC50:  83nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462302(CHEMBL4250215)
Affinity DataEC50:  124nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462289(CHEMBL4245968)
Affinity DataEC50:  37nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462292(CHEMBL4246134)
Affinity DataEC50:  1.00E+5nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462280(CHEMBL4244929)
Affinity DataEC50:  6.20E+3nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462293(CHEMBL4237802)
Affinity DataEC50:  1.27E+4nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462294(CHEMBL4237453)
Affinity DataEC50:  36nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462278(CHEMBL4241613)
Affinity DataEC50:  7.60nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462302(CHEMBL4250215)
Affinity DataEC50:  7.70nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462281(CHEMBL4245391)
Affinity DataEC50:  2.10nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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