Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 50002272
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50021195(2-Hydroxy-ethanesulfonic acid (1,3,4,5,6,11b-hexah...)
Affinity DataKi:  0.770nMAssay Description:Evaluated for its ability to displace [3H]-clonidine from alpha-2 adrenergic receptor of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50021195(2-Hydroxy-ethanesulfonic acid (1,3,4,5,6,11b-hexah...)
Affinity DataKi:  1.10nMAssay Description:Compound was tested for inhibition of human plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50021196(2-Hydroxy-ethanesulfonic acid (1,3,4,5,6,11b-hexah...)
Affinity DataKi:  1.40nMAssay Description:Evaluated for its ability to displace [3H]-clonidine from alpha-2 adrenergic receptor of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50021196(2-Hydroxy-ethanesulfonic acid (1,3,4,5,6,11b-hexah...)
Affinity DataKi:  1.60nMAssay Description:Compound was tested for inhibition of hog kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  10nMAssay Description:Compound was tested for inhibition of hog kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  49nMAssay Description:Evaluated for its ability to displace [3H]-clonidine from alpha-2 adrenergic receptor of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50021197(2-Hydroxy-ethanesulfonic acid (1,3,4,5,6,11b-hexah...)
Affinity DataKi:  100nMAssay Description:Evaluated for its ability to displace [3H]-clonidine from alpha-2 adrenergic receptor of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
TBA

Curated by ChEMBL
LigandPNGBDBM50021195(2-Hydroxy-ethanesulfonic acid (1,3,4,5,6,11b-hexah...)
Affinity DataKi:  110nMAssay Description:Evaluated for its ability to displace [3H]-prazosin from alpha1-Adrenoreceptor of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50021197(2-Hydroxy-ethanesulfonic acid (1,3,4,5,6,11b-hexah...)
Affinity DataKi:  190nMAssay Description:Compound was tested for inhibition of human plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
TBA

Curated by ChEMBL
LigandPNGBDBM50021196(2-Hydroxy-ethanesulfonic acid (1,3,4,5,6,11b-hexah...)
Affinity DataKi:  210nMAssay Description:Evaluated for its ability to displace [3H]-prazosin from alpha1-Adrenoreceptor of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
TBA

Curated by ChEMBL
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  220nMAssay Description:Evaluated for its ability to displace [3H]-prazosin from alpha1-Adrenoreceptor of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
TBA

Curated by ChEMBL
LigandPNGBDBM50021197(2-Hydroxy-ethanesulfonic acid (1,3,4,5,6,11b-hexah...)
Affinity DataKi:  8.00E+3nMAssay Description:Evaluated for its ability to displace [3H]-prazosin from alpha1-Adrenoreceptor of calf cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed