Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50002324
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021422(2,6,6-Trimethyl-bicyclo[3.1.1]heptane-3-carboxylic...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021422(2,6,6-Trimethyl-bicyclo[3.1.1]heptane-3-carboxylic...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021441(2-Phenethyl-benzoic acid 1,4-dimethyl-piperidin-4-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021446(2-Benzyl-benzoic acid 1-methyl-piperidin-4-yl este...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021444(2-Phenoxy-benzoic acid 1-methyl-piperidin-4-yl est...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021438(Biphenyl-2-carboxylic acid 1,4-dimethyl-piperidin-...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021432(2-Phenethyl-benzoic acid 2-diethylamino-ethyl este...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021421(Biphenyl-2-carboxylic acid 3-diethylamino-propyl e...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021439(2-Phenethyl-benzoic acid 1-methyl-piperidin-4-yl e...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021436(2-Phenethyl-benzoic acid 3-diethylamino-propyl est...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021427(Biphenyl-2-carboxylic acid 2-diethylamino-1-methyl...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021428(Biphenyl-2-carboxylic acid 2-diethylamino-ethyl es...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021420(3,4-Dimethoxy-benzoic acid 1-methyl-piperidin-4-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021434(2-Benzoyl-benzoic acid 1-methyl-piperidin-4-yl est...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021425(CHEMBL39641 | Naphthalene-2-carboxylic acid 1-meth...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021424(4-Chloro-benzoic acid 1-methyl-piperidin-4-yl este...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021429(CHEMBL39512 | Propionic acid 1-methyl-piperidin-4-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021426(4-Methyl-benzoic acid 1-methyl-piperidin-4-yl este...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240457(2,4,5-Trimethyl-1H-pyrrole-3-carboxylic acid 1-met...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021430(2,4,5-Trimethyl-benzoic acid 1-methyl-piperidin-4-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021431(2-Bromo-benzoic acid 1-methyl-piperidin-4-yl ester...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021419(2-Methoxy-benzoic acid 1-methyl-piperidin-4-yl est...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021442(2-Phenoxymethyl-benzoic acid 1-methyl-piperidin-4-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021423(3-Hydroxy-benzoic acid 1-methyl-piperidin-4-yl est...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021443(Biphenyl-2-carboxylic acid 1-methyl-piperidin-4-yl...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021440(3-Methoxy-benzoic acid 1-methyl-piperidin-4-yl est...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021437(5-Ethyl-5-phenylbarbituric acid | 5-Phenyl-5-ethyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021445(3-(3,4-Dimethoxy-phenyl)-propionic acid 1-methyl-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021435(Biphenyl-4-carboxylic acid 1-methyl-piperidin-4-yl...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021433(Adamantane-1-carboxylic acid 1,4-dimethyl-piperidi...)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50003655(Phenytoin)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of [3H]-BTX binding to guinea pig voltage-dependent sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed