Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50008343
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518323(CHEMBL4560969)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518339(CHEMBL4514819)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518330(CHEMBL4450254)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518326(CHEMBL4465007)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518331(CHEMBL4582595)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518319(CHEMBL4435935)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518320(CHEMBL4536811)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518338(CHEMBL4576899)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518322(CHEMBL4443245)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518317(CHEMBL4483571)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518315(CHEMBL4581507)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518336(CHEMBL4436378)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518327(CHEMBL4448579)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518329(CHEMBL4585874)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50269809(CHEMBL4077195)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518325(CHEMBL4445334)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518334(CHEMBL4440271)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518333(CHEMBL4467262)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518332(CHEMBL4532879)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518324(CHEMBL4452797)
Affinity DataIC50:  32nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518316(CHEMBL4457647)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518337(CHEMBL4549792)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518321(CHEMBL4443438)
Affinity DataIC50:  40nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518318(CHEMBL4521733)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518335(CHEMBL4547658)
Affinity DataIC50:  63nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518328(CHEMBL4592565)
Affinity DataIC50:  63nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518316(CHEMBL4457647)
Affinity DataIC50:  100nMAssay Description:Inhibition of parkinson's patient-derived LRRK2 G2019S mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518316(CHEMBL4457647)
Affinity DataIC50:  158nMAssay Description:Inhibition of human lymphoblastoid cell-derived LRRK2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518327(CHEMBL4448579)
Affinity DataIC50:  251nMAssay Description:Inhibition of parkinson's patient-derived LRRK2 G2019S mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518327(CHEMBL4448579)
Affinity DataIC50:  398nMAssay Description:Inhibition of human lymphoblastoid cell-derived LRRK2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518316(CHEMBL4457647)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of human CYP3A4 using atorvastatin as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518327(CHEMBL4448579)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of human ERG by IonWork assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518327(CHEMBL4448579)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human CYP3A4 using atorvastatin as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518316(CHEMBL4457647)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518327(CHEMBL4448579)
Affinity DataIC50:  3.98E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518316(CHEMBL4457647)
Affinity DataIC50: <6.31E+4nMAssay Description:Inhibition of human ERG by IonWork assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518327(CHEMBL4448579)
Affinity DataEC50: <5.01E+4nMAssay Description:Activation of human PXRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D

Curated by ChEMBL
LigandPNGBDBM50518316(CHEMBL4457647)
Affinity DataEC50: <5.01E+4nMAssay Description:Activation of human PXRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed