TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of recombinant 6His-Tev-tagged LRRK2 (1326 to 2527) (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotin-RLGRD...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of parkinson's patient-derived LRRK2 G2019S mutantMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Inhibition of human lymphoblastoid cell-derived LRRK2More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of parkinson's patient-derived LRRK2 G2019S mutantMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 398nMAssay Description:Inhibition of human lymphoblastoid cell-derived LRRK2More data for this Ligand-Target Pair
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of human CYP3A4 using atorvastatin as substrateMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of human ERG by IonWork assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP3A4 using atorvastatin as substrateMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataIC50: <6.31E+4nMAssay Description:Inhibition of human ERG by IonWork assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataEC50: <5.01E+4nMAssay Description:Activation of human PXRMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Gsk Pharmaceuticals R&D
Curated by ChEMBL
Affinity DataEC50: <5.01E+4nMAssay Description:Activation of human PXRMore data for this Ligand-Target Pair