Compile Data Set for Download or QSAR
maximum 50k data
Found 37 Enz. Inhib. hit(s) with all data for entry = 50007218
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  180nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of pNP-beta-GlcNAc as substrate by Lineweaver-burk ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)
Affinity DataKi:  190nMAssay Description:Inhibition of human HexBMore data for this Ligand-Target Pair
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507478(CHEMBL4440132)
Affinity DataKi:  600nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507463(CHEMBL4452208)
Affinity DataKi:  700nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507475(CHEMBL4435797)
Affinity DataKi:  800nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507472(CHEMBL4548064)
Affinity DataKi:  900nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507470(CHEMBL4448965)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507462(CHEMBL4548738)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507475(CHEMBL4435797)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507464(CHEMBL4438655)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507463(CHEMBL4452208)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507472(CHEMBL4548064)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507469(CHEMBL4454357)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507470(CHEMBL4448965)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507469(CHEMBL4454357)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507476(CHEMBL4555514)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507461(CHEMBL4592668)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of human beta-N-acetylhexosaminidase using pNP-beta-GlcNAc as substrate by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507462(CHEMBL4548738)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50491601(CHEMBL2333316)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of human beta-N-acetylhexosaminidase using p-nitrophenyl glycoside as substrate by spectrometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507474(CHEMBL4455894)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507471(CHEMBL4540913)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507460(CHEMBL4471966)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate measured after 30 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507460(CHEMBL4471966)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using 4-Mu-GlcNAc as substrate measured after 30 mins by fluorescence as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507476(CHEMBL4555514)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507471(CHEMBL4540913)
Affinity DataKi:  5.10E+3nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507473(CHEMBL4559735)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507477(CHEMBL4564023)
Affinity DataKi:  8.30E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507468(CHEMBL4474777)
Affinity DataKi:  1.59E+4nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507464(CHEMBL4438655)
Affinity DataKi:  2.21E+4nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507468(CHEMBL4474777)
Affinity DataKi:  2.47E+4nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507460(CHEMBL4471966)
Affinity DataKi:  3.04E+4nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate measured after 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507460(CHEMBL4471966)
Affinity DataKi:  3.04E+4nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using 4-Mu-GlcNAc as substrate measured after 30 mins by fluorescence a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507473(CHEMBL4559735)
Affinity DataKi:  5.62E+4nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using varying levels of 4-Mu-GlcNAc as substrate preincubated for 10 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507467(CHEMBL4544229)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human beta-N-acetylhexosaminidase using pNP-beta-GlcNAc as substrate by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507465(CHEMBL4473907)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using 4-Mu-GlcNAc as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507466(CHEMBL4564362)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of recombinant human OGA expressed in Escherichia coli BL21 (DE3) using 4-Mu-GlcNAc as substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-hexosaminidase subunit beta(Homo sapiens (Human))
China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50507466(CHEMBL4564362)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human His6-tagged HexB expressed in Pichia pastoris using 4-Mu-GlcNAc as substrate preincubated for 10 mins followed by sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed