Compile Data Set for Download or QSAR
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Found 64 Enz. Inhib. hit(s) with all data for entry = 50009565
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  46nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPS as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  46nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPS as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  48nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPG as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  48nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free [14C]-AA formation after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  48nMAssay Description:Inhibition of human recombinant iPLA2 assessed as reduction in free FA formation after 30 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  48nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free [14C]-AA formation after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  48nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPG as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  48nMAssay Description:Inhibition of human recombinant iPLA2 assessed as reduction in free FA formation after 30 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  49nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free AA formation after 30 mins by HPLC-MS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  49nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free AA formation after 30 mins by HPLC-MS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  50nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as assessed as reduction in free AA formation after 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  50nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as assessed as reduction in free AA formation after 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  54nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  54nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  55nMAssay Description:Inhibition of human recombinant iPLA2 assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  55nMAssay Description:Inhibition of human recombinant iPLA2 assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  56nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free [14C]-AA formation after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  56nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free [14C]-AA formation after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  63nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  63nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  67nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PLPC as substrate assessed as reduction in free AA formation after 30 mins by HPLC-MS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  67nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PLPC as substrate assessed as reduction in free AA formation after 30 mins by HPLC-MS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  83nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PLPC as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  83nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PLPC as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50529953(CHEMBL4438490)
Affinity DataIC50:  90nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPA as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50529953(CHEMBL4438490)
Affinity DataIC50:  90nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPA as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  104nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  104nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup XIIB secretory phospholipase A2-like protein(Homo sapiens)
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  114nMAssay Description:Inhibition of human recombinant sPLA2 assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup XIIB secretory phospholipase A2-like protein(Homo sapiens)
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  114nMAssay Description:Inhibition of human recombinant sPLA2 assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  131nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free AA formation after 30 mins by HPLC-MS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup XIIB secretory phospholipase A2-like protein(Homo sapiens)
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  131nMAssay Description:Inhibition of human recombinant sPLA2 assessed as reduction in free FA formation after 30 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup XIIB secretory phospholipase A2-like protein(Homo sapiens)
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  131nMAssay Description:Inhibition of human recombinant sPLA2 assessed as reduction in free FA formation after 30 mins by HPLC-MS analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  131nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free AA formation after 30 mins by HPLC-MS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  160nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPA as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371970(CHEMBL89506)
Affinity DataIC50:  160nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPA as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPG as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPG as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  330nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPS as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  330nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPS as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  590nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  590nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as assessed as reduction in free AA formation after 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as assessed as reduction in free AA formation after 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50529953(CHEMBL4438490)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free [14C]-AA formation after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50529953(CHEMBL4438490)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free [14C]-AA formation after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50529953(CHEMBL4438490)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as assessed as reduction in free AA formation after 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50529953(CHEMBL4438490)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as assessed as reduction in free AA formation after 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50529953(CHEMBL4438490)
Affinity DataIC50:  1.39E+3nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PLPC as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50529953(CHEMBL4438490)
Affinity DataIC50:  1.39E+3nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PLPC as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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