Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 50009595
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataKi:  700nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataKi:  700nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530338(CHEMBL1621959)
Affinity DataKi:  1.10E+3nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530338(CHEMBL1621959)
Affinity DataKi:  1.10E+3nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530336(CHEMBL4462082)
Affinity DataKi:  1.60E+3nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530336(CHEMBL4462082)
Affinity DataKi:  1.60E+3nMAssay Description:Mixed-type inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human CLK2 in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human CLK2 in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of recombinant human DYRK1B in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of recombinant human DYRK1B in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of recombinant human DYRK1A in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of recombinant human DYRK1A in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM165207(US8168651, Compound TABLE 16.1 | US9062043, Table ...)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM165207(US8168651, Compound TABLE 16.1 | US9062043, Table ...)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha V73A mutant in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha V73A mutant in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha K74A mutant in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha K74A mutant in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530336(CHEMBL4462082)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530332(CHEMBL4439686)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of CK2alpha (unknown origin) incubated for 40 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530332(CHEMBL4439686)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of CK2alpha (unknown origin) incubated for 40 mins by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530336(CHEMBL4462082)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha H160A mutant in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha H160A mutant in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530338(CHEMBL1621959)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530338(CHEMBL1621959)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha K77A mutant in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530325(CHEMBL4458300)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha K77A mutant in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530318(CHEMBL4526405)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530318(CHEMBL4526405)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530316(CHEMBL4455046)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530316(CHEMBL4455046)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530337(CHEMBL4557432)
Affinity DataIC50:  2.77E+4nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Saarland University

Curated by ChEMBL
LigandPNGBDBM50530337(CHEMBL4557432)
Affinity DataIC50:  2.77E+4nMAssay Description:Inhibition of recombinant human GST-tagged CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed