Found 25 Enz. Inhib. hit(s) with all data for entry = 50007604 Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Inhibition of 5-HT2B receptor (unknown origin)More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: 124nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: 524nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: 650nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: 1.35E+3nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: 4.06E+3nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: 5.69E+3nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: 1.04E+4nMAssay Description:Displacement of [3H]-CCPA binding from human A1 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CCPA binding from human A1 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CCPA binding from human A1 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-NECA from human A2A receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: 4.08E+4nMAssay Description:Displacement of [3H]-CCPA binding from human A1 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]-CCPA binding from human A1 receptor expressed in CHO cells by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin) expressed in baculovirus infected Sf9 insect cells using GST-Rb as substrate in presence of [33P] ATP i...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin) expressed in baculovirus infected Sf9 insect cells using GST-Rb as substrate in presence of [33P] ATP i...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin) expressed in baculovirus infected Sf9 insect cells using GST-Rb as substrate in presence of [33P] ATP i...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected Sf9 insect cells using GST-Rb as substrate in presence of [33P] ATP in...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected Sf9 insect cells using GST-Rb as substrate in presence of [33P] ATP in...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataIC50: 880nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected Sf9 insect cells using GST-Rb as substrate in presence of [33P] ATP in...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataIC50: 2.27E+3nMAssay Description:Inhibition of N-terminal GST-tagged human VEGFR2 (805 to 1356 residues) expressed in a baculovirus infected Sf9 insect cell by Kinase-Glo Plus reagen...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of N-terminal GST-tagged human VEGFR2 (805 to 1356 residues) expressed in a baculovirus infected Sf9 insect cell by Kinase-Glo Plus reagen...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
University Of Science & Technology (Ust)
Curated by ChEMBL
University Of Science & Technology (Ust)
Curated by ChEMBL
Affinity DataIC50: 5.48E+3nMAssay Description:Inhibition of N-terminal GST-tagged human VEGFR2 (805 to 1356 residues) expressed in a baculovirus infected Sf9 insect cell by Kinase-Glo Plus reagen...More data for this Ligand-Target Pair
