Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50007767
Targetvon Hippel-Lindau disease tumor suppressor(Homo sapiens (Human))
Shaoxing University

Curated by ChEMBL
LigandPNGBDBM50246759(CHEMBL4098772)
Affinity DataIC50:  656nMAssay Description:Binding affinity to VHL in human THP-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein cereblon(Homo sapiens (Human))
Shaoxing University

Curated by ChEMBL
LigandPNGBDBM50512415(CHEMBL4226052)
Affinity DataKd:  28nMAssay Description:Binding affinity to CRBN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Shaoxing University

Curated by ChEMBL
LigandPNGBDBM50512415(CHEMBL4226052)
Affinity DataKd:  28nMAssay Description:Binding affinity to BRD4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed