Compile Data Set for Download or QSAR
maximum 50k data
Found 52 Enz. Inhib. hit(s) with all data for entry = 50008845
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50400272(CHEMBL2180727)
Affinity DataIC50:  82nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522839(CHEMBL2095003 | DNDI1417825)
Affinity DataIC50:  410nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522834(CHEMBL4570376)
Affinity DataIC50:  800nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522839(CHEMBL2095003 | DNDI1417825)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522846(CHEMBL4574726)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522838(CHEMBL4451545)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522834(CHEMBL4570376)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522838(CHEMBL4451545)
Affinity DataIC50:  4.76E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522849(CHEMBL4556155)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522846(CHEMBL4574726)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522849(CHEMBL4556155)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522838(CHEMBL4451545)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522842(CHEMBL4456155)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522847(CHEMBL4450318)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522842(CHEMBL4456155)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522849(CHEMBL4556155)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522847(CHEMBL4450318)
Affinity DataIC50:  1.27E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522844(CHEMBL4464973)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522834(CHEMBL4570376)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522844(CHEMBL4464973)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522839(CHEMBL2095003 | DNDI1417825)
Affinity DataIC50:  4.37E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522836(CHEMBL4539487)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522835(CHEMBL4584017)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522837(CHEMBL4524603)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522848(CHEMBL4455478)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522847(CHEMBL4450318)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522848(CHEMBL4455478)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522843(CHEMBL4446512)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522845(CHEMBL4448094)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522841(CHEMBL4558918)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522840(CHEMBL4537226)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522845(CHEMBL4448094)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522837(CHEMBL4524603)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522843(CHEMBL4446512)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522841(CHEMBL4558918)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522840(CHEMBL4537226)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522845(CHEMBL4448094)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522844(CHEMBL4464973)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522843(CHEMBL4446512)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522842(CHEMBL4456155)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522841(CHEMBL4558918)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522840(CHEMBL4537226)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522837(CHEMBL4524603)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522836(CHEMBL4539487)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522835(CHEMBL4584017)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522848(CHEMBL4455478)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522835(CHEMBL4584017)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522836(CHEMBL4539487)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522846(CHEMBL4574726)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Homo sapiens (Human))
Huazhong Agricultural University

Curated by ChEMBL
LigandPNGBDBM50522839(CHEMBL2095003 | DNDI1417825)
Affinity DataKd:  3.80E+3nMAssay Description:Binding affinity to N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in BL21 cells assessed as equilibrium dissociation constant ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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