TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 9.60nMAssay Description:Inhibition of human recombinant BRAF V600E mutant using MEK1 as substrate measured after 1 hr by Western blot analysisMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant BRAF V600E mutant using MEK1 as substrate measured after 1 hr by Western blot analysisMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 92nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 157nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen
Curated by ChEMBL
University Medical Center Groningen
Curated by ChEMBL
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair