Target72 kDa type IV collagenase(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:Inhibition of MMP2 catalytic domain (unknown origin) using Ac-PLG-[2-mercapto-4-methylpentanoyl]-LG-OC2H5 as substrate preincubated for 45 to 120 min...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of COX2 (unknown origin) by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 880nMAssay Description:Inhibition of COX2 (unknown origin) by EIAMore data for this Ligand-Target Pair
TargetLarge neutral amino acids transporter small subunit 1(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Inhibition of recombinant human LAT1More data for this Ligand-Target Pair
TargetProbable maltase-glucoamylase 2(Homo sapiens)
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 2.85E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl alpha-d-glucopyranoside as substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of 5-LOX (unknown origin)More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of 5-LOX (unknown origin)More data for this Ligand-Target Pair
TargetProbable maltase-glucoamylase 2(Homo sapiens)
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataIC50: 8.17E+5nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl alpha-d-glucopyranoside as substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Maharaja Ranjit Singh Punjab Technical University
Curated by ChEMBL
Affinity DataEC50: 5.90E+3nMAssay Description:Inhibition of PPARgamma (unknown origin)More data for this Ligand-Target Pair