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Found 9 Enz. Inhib. hit(s) with all data for entry = 50009408
Target72 kDa type IV collagenase(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University

Curated by ChEMBL
LigandPNGBDBM50528546(CHEMBL4516243)
Affinity DataIC50:  620nMAssay Description:Inhibition of MMP2 catalytic domain (unknown origin) using Ac-PLG-[2-mercapto-4-methylpentanoyl]-LG-OC2H5 as substrate preincubated for 45 to 120 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  840nMAssay Description:Inhibition of COX2 (unknown origin) by EIAMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University

Curated by ChEMBL
LigandPNGBDBM50528543(CHEMBL4540611)
Affinity DataIC50:  880nMAssay Description:Inhibition of COX2 (unknown origin) by EIAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLarge neutral amino acids transporter small subunit 1(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University

Curated by ChEMBL
LigandPNGBDBM50528545(CHEMBL4526588)
Affinity DataIC50:  980nMAssay Description:Inhibition of recombinant human LAT1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProbable maltase-glucoamylase 2(Homo sapiens)
Maharaja Ranjit Singh Punjab Technical University

Curated by ChEMBL
LigandPNGBDBM50502004(CHEMBL4453256)
Affinity DataIC50:  2.85E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl alpha-d-glucopyranoside as substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University

Curated by ChEMBL
LigandPNGBDBM50000541((+-)-1-(1-Benzo[b]thien-2-ylethyl)-1-hydroxyurea |...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of 5-LOX (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University

Curated by ChEMBL
LigandPNGBDBM152734(11-bromo-5-[4-(2-fluorophenyl)piperazine-1- carbon...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of 5-LOX (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable maltase-glucoamylase 2(Homo sapiens)
Maharaja Ranjit Singh Punjab Technical University

Curated by ChEMBL
LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50:  8.17E+5nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl alpha-d-glucopyranoside as substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Maharaja Ranjit Singh Punjab Technical University

Curated by ChEMBL
LigandPNGBDBM50528544(CHEMBL4587922)
Affinity DataEC50:  5.90E+3nMAssay Description:Inhibition of PPARgamma (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed