Affinity DataKi: 0.160nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of activated coagulation factor 11 (unknown origin) assessed as inhibitory constantMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 99nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 175nMAssay Description:Inhibition of activated coagulation factor 11 (unknown origin) assessed as inhibitory constantMore data for this Ligand-Target Pair
Affinity DataKi: 189nMAssay Description:Inhibition of activated coagulation factor 11 (unknown origin) assessed as inhibitory constantMore data for this Ligand-Target Pair
Affinity DataKi: 201nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 333nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 372nMAssay Description:Inhibition of activated coagulation factor 11 (unknown origin) assessed as inhibitory constantMore data for this Ligand-Target Pair
Affinity DataKi: 422nMAssay Description:Inhibition of activated coagulation factor 11 (unknown origin) assessed as inhibitory constantMore data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Inhibition of activated human coagulation factor 11 using pyroGlu-Pro-Arg-pNA as substrate incubated for 10 to 120 mins by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 871nMAssay Description:Inhibition of activated coagulation factor 11 (unknown origin) assessed as inhibitory constantMore data for this Ligand-Target Pair
Affinity DataKi: >3.05E+3nMAssay Description:Inhibition of activated human coagulation factor 12More data for this Ligand-Target Pair
Affinity DataKi: >3.05E+3nMAssay Description:Inhibition of activated human coagulation factor 12More data for this Ligand-Target Pair
Affinity DataKi: 3.66E+3nMAssay Description:Inhibition of activated human coagulation factor 10More data for this Ligand-Target Pair
Affinity DataKi: 4.85E+3nMAssay Description:Inhibition of activated human coagulation factor 7More data for this Ligand-Target Pair
Affinity DataKi: >6.15E+3nMAssay Description:Inhibition of human TPAMore data for this Ligand-Target Pair
Affinity DataKi: >6.15E+3nMAssay Description:Inhibition of human TPAMore data for this Ligand-Target Pair
Affinity DataKi: >6.26E+3nMAssay Description:Inhibition of human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 6.26E+3nMAssay Description:Inhibition of human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: >7.16E+3nMAssay Description:Inhibition of human activated protein CMore data for this Ligand-Target Pair
Affinity DataKi: >9.00E+3nMAssay Description:Inhibition of activated human coagulation factor 10More data for this Ligand-Target Pair
Affinity DataKi: >1.33E+4nMAssay Description:Inhibition of activated coagulation factor 11 (unknown origin) assessed as inhibitory constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.33E+4nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: >1.33E+4nMAssay Description:Inhibition of activated human coagulation factor 7More data for this Ligand-Target Pair
Affinity DataKi: >1.33E+4nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: >1.51E+4nMAssay Description:Inhibition of human urokinaseMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: >1.51E+4nMAssay Description:Inhibition of human urokinaseMore data for this Ligand-Target Pair
Affinity DataKi: >1.52E+4nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
Affinity DataKi: >1.52E+4nMAssay Description:Inhibition of human plasminMore data for this Ligand-Target Pair
Affinity DataKi: >2.15E+4nMAssay Description:Inhibition of human activated protein CMore data for this Ligand-Target Pair
Affinity DataKi: >2.71E+4nMAssay Description:Inhibition of activated human coagulation factor 9More data for this Ligand-Target Pair
Affinity DataKi: >2.71E+4nMAssay Description:Inhibition of activated human coagulation factor 9More data for this Ligand-Target Pair