TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: <1nMAssay Description:Inhibition of His6-tagged MCL1 (unknown origin) incubated for 0.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Inhibition of His6-tagged MCL1 (unknown origin) incubated for 0.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Inhibition of MCL1 (unknown origin)More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Inhibition of His6-tagged MCL1 (unknown origin) incubated for 0.5 hrs in presence of 1% FBS by TR-FRET assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Inhibition of His6-tagged MCL1 (unknown origin) incubated for 0.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 108nMAssay Description:Inhibition of His6-tagged MCL1 (unknown origin) incubated for 0.5 hrs in presence of 1% FBS by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Inhibition of His6-tagged MCL1 (unknown origin) incubated for 0.5 hrs in presence of 1% FBS by TR-FRET assayMore data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of HDAC (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Inhibition of HDAC in human K562 cell extracts using (QSY-7)-RGGRGLGK(Ac)-GGARRHRK(TAMRA)NH2 as substrate preincubated for 30 mins followed by additi...More data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human C-terminal GST/His-tagged HDAC3 (1 to 428 residues) co-expressed with human N-terminal GST-tagged NCOR2 (395 to 489 r...More data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC in human HeLa cell extractsMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibition of HDAC10 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibition of HDAC1 (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 143nMAssay Description:Inhibition of HDAC in human K562 cell extracts using (QSY-7)-RGGRGLGK(Ac)-GGARRHRK(TAMRA)NH2 as substrate preincubated for 30 mins followed by additi...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of bovine brain tubulin polymerization incubated for 1 hrMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of HDAC6 (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of HDAC8 (unknown origin) by fluorescence based assayMore data for this Ligand-Target Pair
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization by spectrometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 8.72E+3nMAssay Description:Inhibition of recombinant human CYP19 using MFC as substrate incubated for 30 mins in presence of NADPH by fluorescence based assayMore data for this Ligand-Target Pair