Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50006758
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503115(CHEMBL4532662)
Affinity DataEC50:  11nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503129(CHEMBL4562979)
Affinity DataEC50:  7.40nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503117(CHEMBL4540607)
Affinity DataEC50:  19nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50469400(CHEMBL4278109)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503118(CHEMBL4515010)
Affinity DataEC50:  12nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503119(CHEMBL4518548)
Affinity DataEC50:  4.40nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503116(CHEMBL4579147)
Affinity DataEC50:  24nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503120(CHEMBL4461571)
Affinity DataEC50:  21nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503121(CHEMBL4544366)
Affinity DataEC50:  3.60nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503122(CHEMBL4470932)
Affinity DataEC50:  13nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503123(CHEMBL4545684)
Affinity DataEC50:  5.30nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503124(CHEMBL4559460)
Affinity DataEC50:  7.30nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503118(CHEMBL4515010)
Affinity DataEC50:  7nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503125(CHEMBL4454228)
Affinity DataEC50:  32nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503120(CHEMBL4461571)
Affinity DataEC50:  3nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503126(CHEMBL4570877)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503121(CHEMBL4544366)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503122(CHEMBL4470932)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503123(CHEMBL4545684)
Affinity DataEC50:  1nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503127(CHEMBL4579525)
Affinity DataEC50:  86nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503125(CHEMBL4454228)
Affinity DataEC50:  32nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503128(CHEMBL4570541)
Affinity DataEC50:  4.20nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503119(CHEMBL4518548)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503115(CHEMBL4532662)
Affinity DataEC50:  2nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503124(CHEMBL4559460)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503126(CHEMBL4570877)
Affinity DataEC50:  19nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503117(CHEMBL4540607)
Affinity DataEC50:  23nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503129(CHEMBL4562979)
Affinity DataEC50:  1nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503128(CHEMBL4570541)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503130(CHEMBL4454138)
Affinity DataEC50:  2.19E+3nMAssay Description:Transactivation of chimeric GAL4-fused human PPARgamma transfected in HEK293EBNA cells measured at 24 hrs after drug treatment by steady-Glo lucifera...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50503116(CHEMBL4579147)
Affinity DataEC50:  22nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed