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Found 11 Enz. Inhib. hit(s) with all data for entry = 50010934
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50205450((S)-7-(3-(aminomethyl)pyrrolidin-1-yl)-1-cycloprop...)
Affinity DataIC50:  120nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50543559(CHEMBL4648309)
Affinity DataIC50:  950nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50543557(CHEMBL4636070)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50543560(CHEMBL4644781)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50543563(CHEMBL4645741)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50543565(CHEMBL4638646)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50543564(CHEMBL4644915)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50543562(CHEMBL4636102)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50543566(CHEMBL4639662)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50543558(CHEMBL4649758)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50543561(CHEMBL4642955)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed