Compile Data Set for Download or QSAR
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Found 16 Enz. Inhib. hit(s) with all data for entry = 50029458
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284727(3-Allyloxycarbonylamino-5-(3-cyclohexyl-propionylo...)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284732(3-Allyloxycarbonylamino-4-oxo-5-phenethylamino-pen...)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284724(3-Allyloxycarbonylamino-4-oxo-5-(3-phenyl-propiony...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284722(3-Allyloxycarbonylamino-4-oxo-5-(3-phenoxy-propion...)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284718(3-Benzyloxycarbonylamino-4-oxo-5-(3-phenyl-propoxy...)
Affinity DataKi:  2.40E+4nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284726(3-Allyloxycarbonylamino-4-oxo-5-(3-phenyl-propylsu...)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281182(3-(2-{2-[2-Acetylamino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataKi:  4.20E+4nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284731(3-Allyloxycarbonylamino-4-oxo-5-(3-phenyl-propylam...)
Affinity DataKi:  6.70E+4nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284723(3-Allyloxycarbonylamino-5-(benzyl-phenethyl-amino)...)
Affinity DataKi:  6.80E+4nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284729(3-Allyloxycarbonylamino-5-(1,2-diphenyl-ethylamino...)
Affinity DataKi:  7.00E+4nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284725(3-Allyloxycarbonylamino-5-benzylcarbamoyloxy-4-oxo...)
Affinity DataKi:  7.40E+4nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284719((S)-3-Allyloxycarbonylamino-4-oxo-5-[(E)-(3-phenyl...)
Affinity DataKi:  9.00E+4nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284721(3-Allyloxycarbonylamino-5-benzylamino-4-oxo-pentan...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284720(3-Allyloxycarbonylamino-4-oxo-8-phenyl-octanoic ac...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284728(3-Allyloxycarbonylamino-5-(methyl-phenethyl-amino)...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCaspase-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284730(3-Allyloxycarbonylamino-5-(benzhydryl-amino)-4-oxo...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of IL-1 beta converting enzyme (ICE) in human blood monocytesMore data for this Ligand-Target Pair
In DepthDetails Article