Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50029461
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284760(1-((3R,5R)-5-Azepan-1-yl-1-methyl-2-oxo-2,3,4,5-te...)
Affinity DataIC50:  6.90nMAssay Description:Inhibitory activity of the compound against Cholecystokinin type B receptor in guinea pig cerebral cortex using [125 I ]- CCK-8 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  8.5nMAssay Description:Inhibitory activity of the compound against Cholecystokinin type B receptor in guinea pig cerebral cortex using [125 I ]- CCK-8 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284759(1-((3R,5S)-5-Azepan-1-yl-1-methyl-2-oxo-2,3,4,5-te...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity of the compound was determined against Cholecystokinin type B receptor in guinea pig cerebral cortex using [125 I ]- CCK-8 as rad...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281723(CHEMBL34335 | [2-Oxo-3-(3-m-tolyl-ureido)-2,3,4,5-...)
Affinity DataIC50:  110nMAssay Description:Inhibitory activity of the compound against Cholecystokinin type B receptor in guinea pig cerebral cortex using [125 I ]- CCK-8 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284759(1-((3R,5S)-5-Azepan-1-yl-1-methyl-2-oxo-2,3,4,5-te...)
Affinity DataIC50:  121nMAssay Description:Inhibitory activity of the compound was determined against Cholecystokinin type A receptor in rat pancreas using [125 I ]- CCK-8 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50284760(1-((3R,5R)-5-Azepan-1-yl-1-methyl-2-oxo-2,3,4,5-te...)
Affinity DataIC50:  646nMAssay Description:Inhibitory activity of the compound against Cholecystokinin type A receptor in rat pancreas using [125 I ]- CCK-8 as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article