Compile Data Set for Download or QSAR
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Found 38 Enz. Inhib. hit(s) with all data for entry = 50029476
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284902((1-{(R)-1-{3-[(E)-2-(4-Cyclobutyl-thiazol-2-yl)-vi...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284902((1-{(R)-1-{3-[(E)-2-(4-Cyclobutyl-thiazol-2-yl)-vi...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284899(CHEMBL287722 | {1-[(R)-3-[2-(1-Hydroxy-1-methyl-et...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284899(CHEMBL287722 | {1-[(R)-3-[2-(1-Hydroxy-1-methyl-et...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284905((1-{(R)-1-{3-[(E)-2-(5,6-Difluoro-benzothiazol-2-y...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284895((1-{(R)-1-{3-[(E)-2-(4-Cyclopentyl-thiazol-2-yl)-v...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284895((1-{(R)-1-{3-[(E)-2-(4-Cyclopentyl-thiazol-2-yl)-v...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284900(CHEMBL288369 | [1-((R)-3-[2-(1-Hydroxy-1-methyl-et...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284890((1-{(R)-1-{3-[(E)-2-(4-Cyclopropyl-thiazol-2-yl)-v...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284890((1-{(R)-1-{3-[(E)-2-(4-Cyclopropyl-thiazol-2-yl)-v...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284907(CHEMBL41620 | [1-((R)-3-[2-(1-Hydroxy-1-methyl-eth...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284893((1-{(R)-1-{3-[(E)-2-(4-tert-Butyl-thiazol-2-yl)-vi...)
Affinity DataIC50:  2nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284893((1-{(R)-1-{3-[(E)-2-(4-tert-Butyl-thiazol-2-yl)-vi...)
Affinity DataIC50:  2nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284896((1-{(R)-1-{3-[(E)-2-(4-Cyclohexyl-thiazol-2-yl)-vi...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284903((1-{(R)-1-{3-[(E)-2-(5,6-Dihydro-4H-cyclopentathia...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284903((1-{(R)-1-{3-[(E)-2-(5,6-Dihydro-4H-cyclopentathia...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284901((1-{(R)-1-{3-[(E)-2-(5-Fluoro-benzothiazol-2-yl)-v...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50013920(3-[(R)-{3-[(E)-2-(7-Chloro-quinolin-2-yl)-vinyl]-p...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284888((1-{(R)-1-(3-{(E)-2-[4-(4-Fluoro-phenyl)-thiazol-2...)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284888((1-{(R)-1-(3-{(E)-2-[4-(4-Fluoro-phenyl)-thiazol-2...)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284886(CHEMBL41395 | [1-((R)-3-[2-(1-Hydroxy-1-methyl-eth...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284886(CHEMBL41395 | [1-((R)-3-[2-(1-Hydroxy-1-methyl-eth...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284904((1-{(R)-1-{3-[(E)-2-(5-Chloro-benzothiazol-2-yl)-v...)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284904((1-{(R)-1-{3-[(E)-2-(5-Chloro-benzothiazol-2-yl)-v...)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284887(CHEMBL42520 | [1-((R)-3-[2-(1-Hydroxy-1-methyl-eth...)
Affinity DataIC50:  11nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284887(CHEMBL42520 | [1-((R)-3-[2-(1-Hydroxy-1-methyl-eth...)
Affinity DataIC50:  11nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284897(CHEMBL40992 | [1-((R)-3-[2-(1-Hydroxy-1-methyl-eth...)
Affinity DataIC50:  12.8nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284897(CHEMBL40992 | [1-((R)-3-[2-(1-Hydroxy-1-methyl-eth...)
Affinity DataIC50:  13nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284908((1-{(R)-1-[3-((E)-2-Benzothiazol-2-yl-vinyl)-pheny...)
Affinity DataIC50:  17nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284906(CHEMBL40686 | [1-((R)-3-[2-(1-Hydroxy-1-methyl-eth...)
Affinity DataIC50:  42nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284898(CHEMBL42410 | [1-((R)-3-[2-(1-Hydroxy-1-methyl-eth...)
Affinity DataIC50:  48nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284891((1-{(R)-1-(3-{(E)-2-[4-(4-Chloro-phenyl)-thiazol-2...)
Affinity DataIC50:  79nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284891((1-{(R)-1-(3-{(E)-2-[4-(4-Chloro-phenyl)-thiazol-2...)
Affinity DataIC50:  79.3nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284889(CHEMBL40836 | {1-[(R)-3-[2-(1-Hydroxy-1-methyl-eth...)
Affinity DataIC50:  98.7nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284889(CHEMBL40836 | {1-[(R)-3-[2-(1-Hydroxy-1-methyl-eth...)
Affinity DataIC50:  99nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284892((1-{(R)-1-{3-[(E)-2-(5-Chloro-4-isopropyl-thiazol-...)
Affinity DataIC50:  170nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284892((1-{(R)-1-{3-[(E)-2-(5-Chloro-4-isopropyl-thiazol-...)
Affinity DataIC50:  170nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50284894((1-{(R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50:  381nMAssay Description:Inhibition of [3H]-LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In DepthDetails Article