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Found 20 Enz. Inhib. hit(s) with all data for entry = 50029726
TargetSodium- and chloride-dependent GABA transporter 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50003634(1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...)
Affinity DataIC50:  130nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403566(CHEMBL2094022)
Affinity DataIC50:  2.70E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403564(CHEMBL2094024)
Affinity DataIC50:  2.70E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent betaine transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403563(CHEMBL2093977)
Affinity DataIC50:  3.35E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human BGT-1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent betaine transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403564(CHEMBL2094024)
Affinity DataIC50:  4.36E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human BGT-1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50403565(CHEMBL2093978)
Affinity DataIC50:  4.47E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporteMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003634(1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...)
Affinity DataIC50:  5.50E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporteMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403565(CHEMBL2093978)
Affinity DataIC50:  6.32E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50403566(CHEMBL2094022)
Affinity DataIC50:  6.69E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporteMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50403563(CHEMBL2093977)
Affinity DataIC50:  7.57E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporteMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403566(CHEMBL2094022)
Affinity DataIC50:  7.82E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-3 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent betaine transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403566(CHEMBL2094022)
Affinity DataIC50:  8.09E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human BGT-1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403563(CHEMBL2093977)
Affinity DataIC50:  8.09E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 2(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50403564(CHEMBL2094024)
Affinity DataIC50:  8.10E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporteMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403563(CHEMBL2093977)
Affinity DataIC50:  8.76E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-3 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50003634(1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...)
Affinity DataIC50:  9.44E+5nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-3 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403565(CHEMBL2093978)
Affinity DataIC50:  2.04E+6nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-3 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent betaine transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403565(CHEMBL2093978)
Affinity DataIC50:  2.90E+6nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human BGT-1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent GABA transporter 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403564(CHEMBL2094024)
Affinity DataIC50:  3.23E+6nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human GAT-3 transporterMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium- and chloride-dependent betaine transporter(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50003634(1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...)
Affinity DataIC50:  7.21E+6nMAssay Description:Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned human BGT-1 transporterMore data for this Ligand-Target Pair
In DepthDetails Article