Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50029780
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287790((2S,4R)-1-Acetyl-4-benzyloxy-pyrrolidine-2-carboxy...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287780((S)-1-((R)-2-Amino-3-phenyl-propionyl)-pyrrolidine...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287791((2S,4R)-1-((R)-2-Amino-3-phenyl-propionyl)-4-benzy...)
Affinity DataIC50:  3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287788((2S,4R)-1-Acetyl-4-cyclohexylmethoxy-pyrrolidine-2...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287781((2S,4S)-1-((R)-2-Amino-3-phenyl-propionyl)-4-benzy...)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287793((2S,4R)-1-Acetyl-4-(3,3-diphenyl-propoxy)-pyrrolid...)
Affinity DataIC50:  10nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287783((2S,4R)-4-Benzyloxy-1-propionyl-pyrrolidine-2-carb...)
Affinity DataIC50:  13nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287789((2S,4R)-1-Acetyl-4-(3-phenyl-propoxy)-pyrrolidine-...)
Affinity DataIC50:  14nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287794((2S,4R)-1-Acetyl-4-butoxy-pyrrolidine-2-carboxylic...)
Affinity DataIC50:  22nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287787((2S,4R)-4-Benzyloxy-1-methanesulfonyl-pyrrolidine-...)
Affinity DataIC50:  24nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287782((2S,4R)-4-Benzyloxy-1-(3-phenyl-propionyl)-pyrroli...)
Affinity DataIC50:  32nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287792((2S,4R)-1-Acetyl-4-phenethyl-pyrrolidine-2-carboxy...)
Affinity DataIC50:  40nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287786((S)-1-Acetyl-pyrrolidine-2-carboxylic acid [(S)-1-...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287785((2S,4S)-1-Acetyl-4-benzyloxy-pyrrolidine-2-carboxy...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287784((2S,4R)-4-Benzyloxy-1-ethyl-pyrrolidine-2-carboxyl...)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails Article