Affinity DataIC50: 900nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Compound was tested for inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Compound was tested for its ability to inhibit Endothelin A receptor induced arachidonic acid release(AARA) in rabbit renal artery vascular smooth mu...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Compound was tested for its ability to inhibit Endothelin A receptor induced arachidonic acid release(AARA) in rabbit renal artery vascular smooth mu...More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Compound was tested for its ability to inhibit Endothelin A receptor induced arachidonic acid release(AARA) in rabbit renal artery vascular smooth mu...More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Compound was tested for its ability to inhibit Endothelin A receptor induced arachidonic acid release(AARA) in rabbit renal artery vascular smooth mu...More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of binding of [125I]-ET-1 to cloned human Endothelin A receptor expressed in LtK- cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Antagonistic activity against endothelin A receptor in rabbit renal artery vascular smooth muscle cells.More data for this Ligand-Target Pair