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maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50029857
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288748((S)-4-(4-Methoxy-benzenesulfonylamino)-2-[(S)-1-((...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288759((S)-2-[(S)-1-((S)-3-Methyl-1-phenylcarbamoyl-butyl...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50040594((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
Affinity DataIC50:  90nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288758((S)-2-[(S)-1-((S)-1-Methylcarbamoyl-2-phenyl-ethyl...)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50057083((R)-2-((S)-1-((S)-4-methyl-1-oxo-1-(phenylamino)pe...)
Affinity DataIC50:  320nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288752((S)-2-[(S)-1-((S)-1-Methylcarbamoyl-2-phenyl-ethyl...)
Affinity DataIC50:  510nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288756((S)-2-[(S)-1-((S)-1-Benzyloxycarbamoyl-3-methyl-bu...)
Affinity DataIC50:  550nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288749((S)-4-[(1H-Indole-2-carbonyl)-amino]-2-[(S)-1-((S)...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288760((S)-4-(2,4-Dioxo-1,3-diaza-spiro[4.4]non-3-yl)-2-[...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288755(4-({(S)-2-[(S)-1-Carboxy-3-(4-methoxy-benzenesulfo...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288757((S)-4-(4-Methoxy-benzenesulfonylamino)-2-[(S)-1-(4...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288753(4-{(S)-2-[(S)-1-Carboxy-3-(4-methoxy-benzenesulfon...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288751((S)-2-[(S)-1-(4-Methanesulfonyl-piperazine-1-carbo...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288750((S)-2-[(S)-1-(4-Hydroxy-piperidine-1-carbonyl)-3-p...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288761((S)-4-(4-Methoxy-benzenesulfonylamino)-2-[(S)-1-(m...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288754(4-{(S)-2-[(S)-1-Carboxy-3-(4-methoxy-benzenesulfon...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against Matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails Article