Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50034816
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)
Affinity DataKi:  18nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286239(CHEMBL315927 | [(1S,4R,5R)-11-((S)-Isobutyl)-14-((...)
Affinity DataKi:  224nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286244(CHEMBL87296 | [(1S,4R,5R)-8-Benzyl-11-((S)-isobuty...)
Affinity DataKi:  2.40E+3nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286238(CHEMBL314364 | {8-[(1H-Indole-2-carbonyl)-amino]-1...)
Affinity DataKi:  6.00E+3nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286234(CHEMBL86489 | [8-(2-1H-Indol-3-yl-acetylamino)-11-...)
Affinity DataKi:  7.00E+3nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)
Affinity DataKi:  7.00E+3nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286237(CHEMBL86581 | [8-(Naphthalen-1-ylmethoxy)-11-oxo-5...)
Affinity DataKi:  7.00E+3nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286243(CHEMBL421349 | [8-(Naphthalen-1-ylmethoxy)-11-oxo-...)
Affinity DataKi:  8.00E+3nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286240(CHEMBL314915 | {8-[(Naphthalen-1-ylmethyl)-amino]-...)
Affinity DataKi:  9.00E+3nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286242(CHEMBL315096 | {8-[(1H-Indole-3-carbonyl)-amino]-1...)
Affinity DataKi:  1.10E+4nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286235(CHEMBL313184 | [8-(1H-Indol-3-ylmethyl)-11-oxo-5-p...)
Affinity DataKi:  1.20E+4nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286234(CHEMBL86489 | [8-(2-1H-Indol-3-yl-acetylamino)-11-...)
Affinity DataKi:  1.40E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286240(CHEMBL314915 | {8-[(Naphthalen-1-ylmethyl)-amino]-...)
Affinity DataKi:  1.70E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286243(CHEMBL421349 | [8-(Naphthalen-1-ylmethoxy)-11-oxo-...)
Affinity DataKi:  2.80E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286238(CHEMBL314364 | {8-[(1H-Indole-2-carbonyl)-amino]-1...)
Affinity DataKi:  3.30E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286235(CHEMBL313184 | [8-(1H-Indol-3-ylmethyl)-11-oxo-5-p...)
Affinity DataKi:  4.10E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286237(CHEMBL86581 | [8-(Naphthalen-1-ylmethoxy)-11-oxo-5...)
Affinity DataKi:  6.00E+4nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286242(CHEMBL315096 | {8-[(1H-Indole-3-carbonyl)-amino]-1...)
Affinity DataKi:  8.00E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286236(CHEMBL316247 | {8-[(Naphthalene-1-carbonyl)-amino]...)
Affinity DataKi:  8.30E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286241((8-Benzyloxy-11-oxo-5,11-dihydro-dibenzo[b,e][1,4]...)
Affinity DataKi: >1.00E+5nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286241((8-Benzyloxy-11-oxo-5,11-dihydro-dibenzo[b,e][1,4]...)
Affinity DataKi:  1.09E+5nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In DepthDetails Article