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Found 15 Enz. Inhib. hit(s) with all data for entry = 50034901
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50017659(2-(Dimethylamino)ethyl p-(butylamino)benzoate | 2-...)
Affinity DataIC50:  400nMAssay Description:Antagonism of batrachotoxin-mediated sodium ion uptake into cultured neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290406(Benzoic acid 3-dimethylaminomethyl-5-hydroxy-5-(1-...)
Affinity DataIC50:  500nMAssay Description:Antagonism of batrachotoxin-mediated sodium ion uptake into cultured neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290406(Benzoic acid 3-dimethylaminomethyl-5-hydroxy-5-(1-...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of [3H]batrachotoxin binding to rat brain neuronal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290405(1-(1-Benzyloxy-8-methyl-2-oxa-tricyclo[5.3.1.0*3,8...)
Affinity DataIC50:  4.00E+3nMAssay Description:Antagonism of batrachotoxin-mediated sodium ion uptake into cultured neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290405(1-(1-Benzyloxy-8-methyl-2-oxa-tricyclo[5.3.1.0*3,8...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of [3H]batrachotoxin binding to rat brain neuronal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290404(Benzoic acid 5-hydroxy-3-methoxymethyl-5-(1-methox...)
Affinity DataIC50:  5.00E+3nMAssay Description:Antagonism of batrachotoxin-mediated sodium ion uptake into cultured neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50017659(2-(Dimethylamino)ethyl p-(butylamino)benzoate | 2-...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of [3H]batrachotoxin binding to rat brain neuronal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290404(Benzoic acid 5-hydroxy-3-methoxymethyl-5-(1-methox...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of [3H]batrachotoxin binding to rat brain neuronal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290408(CHEMBL298513 | [1-(3-Bromo-benzyloxy)-8-methyl-2-o...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of [3H]batrachotoxin binding to rat brain neuronal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50214776(CHEBI:28051 | VERATRIDINE)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of [3H]batrachotoxin binding to rat brain neuronal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290408(CHEMBL298513 | [1-(3-Bromo-benzyloxy)-8-methyl-2-o...)
Affinity DataIC50:  8.00E+4nMAssay Description:Antagonism of batrachotoxin-mediated sodium ion uptake into cultured neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290407(4-Dimethylamino-1-(1-methoxy-8-methyl-2-oxa-tricyc...)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition of [3H]batrachotoxin binding to rat brain neuronal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290407(4-Dimethylamino-1-(1-methoxy-8-methyl-2-oxa-tricyc...)
Affinity DataIC50:  2.00E+5nMAssay Description:Antagonism of batrachotoxin-mediated sodium ion uptake into cultured neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290403((1-Methoxy-8-methyl-2-oxa-tricyclo[5.3.1.0*3,8*]un...)
Affinity DataIC50:  1.00E+6nMAssay Description:Antagonism of batrachotoxin-mediated sodium ion uptake into cultured neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50290403((1-Methoxy-8-methyl-2-oxa-tricyclo[5.3.1.0*3,8*]un...)
Affinity DataIC50:  2.00E+6nMAssay Description:Inhibition of [3H]batrachotoxin binding to rat brain neuronal membranesMore data for this Ligand-Target Pair
In DepthDetails Article