Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50048636
LigandPNGBDBM50224275(CHEMBL278717)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224275(CHEMBL278717)
Affinity DataIC50:  8nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataIC50:  14nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224274(CHEMBL2304423)
Affinity DataIC50:  16nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224274(CHEMBL2304423)
Affinity DataIC50:  18nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224277(CHEMBL280309)
Affinity DataIC50:  22nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataIC50:  22nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224277(CHEMBL280309)
Affinity DataIC50:  26nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataIC50:  44nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224276(CHEMBL277122)
Affinity DataIC50:  55nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224276(CHEMBL277122)
Affinity DataIC50:  90nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataIC50:  150nMAssay Description:Inhibition of stereospecific [3H]diprenorphine binding to opioid receptors of rat brain homogenates by 50% in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed