Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50005129
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033139(CHEMBL2370495 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*...)
Affinity DataIC50:  0.240nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453783(CHEMBL2311023)
Affinity DataIC50:  0.550nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033143(CHEMBL216640 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*-...)
Affinity DataIC50:  0.580nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453785(CHEMBL2311025)
Affinity DataIC50:  0.610nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453785(CHEMBL2311025)
Affinity DataIC50:  0.640nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453782(CHEMBL2370497)
Affinity DataIC50:  0.900nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033142(CHEMBL2370496 | H-Tyr-Gly-Gly-Phe-Leu-Lys*-Arg*-Il...)
Affinity DataIC50:  4nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033142(CHEMBL2370496 | H-Tyr-Gly-Gly-Phe-Leu-Lys*-Arg*-Il...)
Affinity DataIC50:  4nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033139(CHEMBL2370495 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*...)
Affinity DataIC50:  5.20nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453784(CHEMBL2311024)
Affinity DataIC50:  8nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453782(CHEMBL2370497)
Affinity DataIC50:  9nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033141(CHEMBL2370494 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys*-Ile...)
Affinity DataIC50:  9.20nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033143(CHEMBL216640 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*-...)
Affinity DataIC50:  9.90nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453783(CHEMBL2311023)
Affinity DataIC50:  12nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033142(CHEMBL2370496 | H-Tyr-Gly-Gly-Phe-Leu-Lys*-Arg*-Il...)
Affinity DataIC50:  13nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033141(CHEMBL2370494 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys*-Ile...)
Affinity DataIC50:  17nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033141(CHEMBL2370494 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys*-Ile...)
Affinity DataIC50:  17nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033139(CHEMBL2370495 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*...)
Affinity DataIC50:  18nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453783(CHEMBL2311023)
Affinity DataIC50:  24nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033143(CHEMBL216640 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Ile*-...)
Affinity DataIC50:  26nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453785(CHEMBL2311025)
Affinity DataIC50:  32nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453782(CHEMBL2370497)
Affinity DataIC50:  53nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453784(CHEMBL2311024)
Affinity DataIC50:  96nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453784(CHEMBL2311024)
Affinity DataIC50:  198nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033137(CHEMBL2311022 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-...)
Affinity DataIC50:  1.04E+3nMAssay Description:Binding affinity against Opioid receptor mu 1 from Guinea pig brain homogenate using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033137(CHEMBL2311022 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-...)
Affinity DataIC50:  7.99E+3nMAssay Description:Binding affinity against Opioid receptor kappa 1 of Guinea pig brain homogenate using [3H]U-69,593More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50033137(CHEMBL2311022 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Binding affinity against delta opioid receptor of Guinea pig brain homogenate using [3H]c[D-Pen2,p-Cl-Phe4,D-Pen5]enkephalinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed