Compile Data Set for Download or QSAR
maximum 50k data
Found 57 Enz. Inhib. hit(s) with all data for entry = 50005998
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043582(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-3-p...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of rabbit fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043591(1N-phenyl-11-amino-2-[1-[1-amino-(1R)-ethylcarboxa...)
Affinity DataKi:  110nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043582(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-3-p...)
Affinity DataKi:  200nMpH: 7.5Assay Description:Inhibition of human fibroblast gelatinase A at pH 7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043584(1N-(4-methoxyphenyl)-2-[1-[1-amino-(1R)-ethylcarbo...)
Affinity DataKi:  230nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043593(1N-phenyl-8-amino-2-[1-[1-amino-(1R)-ethylcarboxam...)
Affinity DataKi:  370nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043593(1N-phenyl-8-amino-2-[1-[1-amino-(1R)-ethylcarboxam...)
Affinity DataKi:  370nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043582(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-3-p...)
Affinity DataKi:  410nMAssay Description:Inhibition of rabbit fibroblast gelatinase AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043582(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-3-p...)
Affinity DataKi:  450nMAssay Description:Inhibition of human fibroblast gelatinase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043582(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-3-p...)
Affinity DataKi:  470nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043601(1N-phenyl-7-amino-2-[1-[1-amino-(1R)-ethylcarboxam...)
Affinity DataKi:  510nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043592(1N-(3-methoxyphenyl)-2-[1-[1-amino-(1R)-ethylcarbo...)
Affinity DataKi:  590nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043589(1N-phenyl-6-amino-2-[1-[1-amino-(1R)-ethylcarboxam...)
Affinity DataKi:  640nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043582(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-3-p...)
Affinity DataKi:  760nMpH: 6.5Assay Description:Inhibition of human fibroblast collagenase at pH 6.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043582(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-3-p...)
Affinity DataKi:  760nMAssay Description:Inhibition of rabbit fibroblast gelatinase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043596(1N-phenyl-4-amino-2-[1-[1-amino-(1R)-ethylcarboxam...)
Affinity DataKi:  820nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043596(1N-phenyl-4-amino-2-[1-[1-amino-(1R)-ethylcarboxam...)
Affinity DataKi:  820nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043589(1N-phenyl-6-amino-2-[1-[1-amino-(1R)-ethylcarboxam...)
Affinity DataKi:  850nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043591(1N-phenyl-11-amino-2-[1-[1-amino-(1R)-ethylcarboxa...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043592(1N-(3-methoxyphenyl)-2-[1-[1-amino-(1R)-ethylcarbo...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043584(1N-(4-methoxyphenyl)-2-[1-[1-amino-(1R)-ethylcarbo...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043601(1N-phenyl-7-amino-2-[1-[1-amino-(1R)-ethylcarboxam...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043586(1N-phenyl-2-{1-[1-amino-(1R)-ethylcarboxamido]-4-p...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043586(1N-phenyl-2-{1-[1-amino-(1R)-ethylcarboxamido]-4-p...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043600(1N-(2-amino-1-phenylcarbamoylethyl)-2-[1-amino-(1R...)
Affinity DataKi:  3.18E+3nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043590(1N-phenyl-4-amino-2-[1-[1-amino-(1R)-ethylcarboxam...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043590(1N-phenyl-4-amino-2-[1-[1-amino-(1R)-ethylcarboxam...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043594(1N-(2-methoxyphenyl)-2-[1-[1-amino-(1R)-ethylcarbo...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043600(1N-(2-amino-1-phenylcarbamoylethyl)-2-[1-amino-(1R...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043594(1N-(2-methoxyphenyl)-2-[1-[1-amino-(1R)-ethylcarbo...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043578(1N-phenyl-2-[1-amino-(1R)-ethylcarboxamido(phenyl)...)
Affinity DataKi:  3.40E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043582(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-3-p...)
Affinity DataIC50:  61nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043582(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-3-p...)
Affinity DataIC50:  320nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043581(1N-[1-[1-benzylcarbamoyl-2-phenyl-(1S)-ethylcarbam...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043587(1N-[1-benzylcarbamoyl-2-phenyl-(1S)-ethyl]-2-[1-am...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043578(1N-phenyl-2-[1-amino-(1R)-ethylcarboxamido(phenyl)...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043585(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-2-(...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043588(1N-[1-phenyl-(1S)-ethyl]-2-[1-[1-amino-(1R)-ethylc...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043585(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-2-(...)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043581(1N-[1-[1-benzylcarbamoyl-2-phenyl-(1S)-ethylcarbam...)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043588(1N-[1-phenyl-(1S)-ethyl]-2-[1-[1-amino-(1R)-ethylc...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043580(1N-phenethyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-...)
Affinity DataIC50:  1.78E+4nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043578(1N-phenyl-2-[1-amino-(1R)-ethylcarboxamido(phenyl)...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043599(1N-[1-[1-carbamoyl-(1S)-pentylcarbamoyl]-3-methyl-...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043583(1N-benzyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-2-(...)
Affinity DataIC50:  2.39E+4nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043579(1N-[1-carbamoyl-3-methyl-(1S)-butyl]-2-[1-[1-amino...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043597(1N-[1-[1-benzylcarbamoyl-3-methyl-(1S)-butylcarbam...)
Affinity DataIC50:  2.73E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043583(1N-benzyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-2-(...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043580(1N-phenethyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-...)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043602(1N-[1-phenyl-(1R)-ethyl]-2-[1-[1-amino-(1R)-ethylc...)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of human fibroblast stromelysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043595(1N-phenyl-2-[1-[1-amino-(1R)-ethylcarboxamido]-2-p...)
Affinity DataIC50:  5.21E+4nMAssay Description:Inhibition of human fibroblast collagenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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