TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 4.40E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 4.40E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:SKCa-blocking activity as inhibitino of after hyperpolarization (AHP) in cultured rat sympathetic neurons; No activity at maximal dose usedMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:SKCa-blocking activity as inhibition of after hyperpolarization (AHP) in cultured rat sympathetic neurons; Insufficient activity at maximal dose usedMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 1/2/3(Rattus norvegicus)
University College London
Curated by ChEMBL
University College London
Curated by ChEMBL
Affinity DataIC50: 4.00E+4nMAssay Description:SKCa-blocking activity by its ability to inhibit after hyperpolarization (AHP) in cultured rat sympathetic neuronsMore data for this Ligand-Target Pair