Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50006616
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051751(1-[3-(4-Isopropenyl-phenyl)-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051753(1-(3-Naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-yl)...)
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051757(1-[3-(4-Vinyl-phenyl)-8-aza-bicyclo[3.2.1]oct-2-yl...)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50041293(1-(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]...)
Affinity DataKi:  0.390nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051750(1-[3-(4-Isopropenyl-phenyl)-8-methyl-8-aza-bicyclo...)
Affinity DataKi:  0.820nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50041293(1-(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051754(1-[8-Methyl-3-(4-vinyl-phenyl)-8-aza-bicyclo[3.2.1...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051758(1-[3-(4-Isopropyl-phenyl)-8-aza-bicyclo[3.2.1]oct-...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051752(1-(3-p-Tolyl-8-aza-bicyclo[3.2.1]oct-2-yl)-propan-...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051757(1-[3-(4-Vinyl-phenyl)-8-aza-bicyclo[3.2.1]oct-2-yl...)
Affinity DataKi:  10.9nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051752(1-(3-p-Tolyl-8-aza-bicyclo[3.2.1]oct-2-yl)-propan-...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50041303(1-[3-(4-Isopropyl-phenyl)-8-methyl-8-aza-bicyclo[3...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051754(1-[8-Methyl-3-(4-vinyl-phenyl)-8-aza-bicyclo[3.2.1...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051749(1-[3-(4-Cyclohexyl-phenyl)-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051751(1-[3-(4-Isopropenyl-phenyl)-8-aza-bicyclo[3.2.1]oc...)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051755(1-[3-(4-Cyclohexyl-phenyl)-8-methyl-8-aza-bicyclo[...)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50041296(1-(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oct-2-yl...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051756(1-{3-[4-(1-Ethyl-propyl)-phenyl]-8-aza-bicyclo[3.2...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051758(1-[3-(4-Isopropyl-phenyl)-8-aza-bicyclo[3.2.1]oct-...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50041296(1-(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oct-2-yl...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051753(1-(3-Naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-yl)...)
Affinity DataKi:  440nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051759(1-{3-[4-(1-Ethyl-propyl)-phenyl]-8-methyl-8-aza-bi...)
Affinity DataKi:  540nMAssay Description:Displacement of [3H]-paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051750(1-[3-(4-Isopropenyl-phenyl)-8-methyl-8-aza-bicyclo...)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051749(1-[3-(4-Cyclohexyl-phenyl)-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051756(1-{3-[4-(1-Ethyl-propyl)-phenyl]-8-aza-bicyclo[3.2...)
Affinity DataKi:  5.10E+3nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50041303(1-[3-(4-Isopropyl-phenyl)-8-methyl-8-aza-bicyclo[3...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051759(1-{3-[4-(1-Ethyl-propyl)-phenyl]-8-methyl-8-aza-bi...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051755(1-[3-(4-Cyclohexyl-phenyl)-8-methyl-8-aza-bicyclo[...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-nisoxatine from Norepinephrine transporter of rat forebrain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50041293(1-(8-Methyl-3-naphthalen-2-yl-8-aza-bicyclo[3.2.1]...)
Affinity DataIC50:  0.120nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051754(1-[8-Methyl-3-(4-vinyl-phenyl)-8-aza-bicyclo[3.2.1...)
Affinity DataIC50:  0.900nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051757(1-[3-(4-Vinyl-phenyl)-8-aza-bicyclo[3.2.1]oct-2-yl...)
Affinity DataIC50:  1.5nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051752(1-(3-p-Tolyl-8-aza-bicyclo[3.2.1]oct-2-yl)-propan-...)
Affinity DataIC50:  4.70nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051750(1-[3-(4-Isopropenyl-phenyl)-8-methyl-8-aza-bicyclo...)
Affinity DataIC50:  7.20nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50041296(1-(8-Methyl-3-p-tolyl-8-aza-bicyclo[3.2.1]oct-2-yl...)
Affinity DataIC50:  8.20nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051751(1-[3-(4-Isopropenyl-phenyl)-8-aza-bicyclo[3.2.1]oc...)
Affinity DataIC50:  16nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051753(1-(3-Naphthalen-2-yl-8-aza-bicyclo[3.2.1]oct-2-yl)...)
Affinity DataIC50:  36nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051756(1-{3-[4-(1-Ethyl-propyl)-phenyl]-8-aza-bicyclo[3.2...)
Affinity DataIC50:  190nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051759(1-{3-[4-(1-Ethyl-propyl)-phenyl]-8-methyl-8-aza-bi...)
Affinity DataIC50:  270nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051755(1-[3-(4-Cyclohexyl-phenyl)-8-methyl-8-aza-bicyclo[...)
Affinity DataIC50:  320nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50041303(1-[3-(4-Isopropyl-phenyl)-8-methyl-8-aza-bicyclo[3...)
Affinity DataIC50:  440nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051749(1-[3-(4-Cyclohexyl-phenyl)-8-aza-bicyclo[3.2.1]oct...)
Affinity DataIC50:  490nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
State University Of New York

Curated by ChEMBL
LigandPNGBDBM50051758(1-[3-(4-Isopropyl-phenyl)-8-aza-bicyclo[3.2.1]oct-...)
Affinity DataIC50:  540nMAssay Description:Displacement of [125I]-RTI-55 from dopamine transporter of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed