Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50006828
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM2581(3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^...)
Affinity DataIC50:  2.45E+3nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054428(13-(3,4-dihydroxy-6-hydroxymethyl-5-methoxytetrahy...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054426(7-hydroxy-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)
Affinity DataIC50:  2.21E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054423(1,11-dichloro-13-(3,4-dihydroxy-6-hydroxymethyl-5-...)
Affinity DataIC50:  2.88E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054429(6-Hydroxy-12-(4-O-methyl-beta-D-glucopyrannosyl) -...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054425(6-amino-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrro...)
Affinity DataIC50:  4.35E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM2672(3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^...)
Affinity DataIC50:  4.47E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054432(1,11-Dichloro-6-hydroxy-12-(4-O-methyl-beta-D-gluc...)
Affinity DataIC50:  6.80E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054434(6-(4-Semicarbazido)-6,7,12,13-tetrahydro-5,7-dioxo...)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054422(6-hydroxy-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)
Affinity DataIC50:  7.92E+4nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054418(1,11-dichloro-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054437(6-Amino-1,11-dichloro-12-(4-O-methyl-beta-D-glucop...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054419(1,11-dichloro-7-hydroxy-6,7,12,13-tetrahydro-5H-in...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054420(12-(3,4-dihydroxy-6-hydroxymethyl-5-methoxytetrahy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054433(6-(2-Hydroxyethyl)6,7,12,13-tetrahydro-5,7-dioxoin...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054435(6-Amino-1,11-dichloro-6,7,12,13-tetrahydro-5,7-dio...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054421(1,11-dichloro-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054436(6-Formamido-6,7,12,13-tetrahydro-5,7-dioxoindolo[2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50162287((Rebeccamycin)1,11-dichloro-12-(3,4-dihydroxy-6-hy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054438(6-Amino-12-(4-O-methyl-beta-D-glucopyrannosyl) -6,...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054431(6-Formamido-12-(4-O-methyl-beta-D-glucopyrannosyl)...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054430(1,11-Dichloro-6-formamido-12-(4-O-methyl-beta-D-gl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50054427(6-Formamido-1,11-dichloro-6,7,12,13-tetrahydro-5,7...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Protein Kinase C(PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed