TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.0150nMAssay Description:Apparent binding affinity against estradiol-stimulated T-47D cell proliferationMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.0160nMAssay Description:Apparent binding affinity against estradiol-stimulated T-47D cell proliferationMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.0230nMAssay Description:Stimulation of alkaline phosphatase activity in human endometrial Ishikawa cells with 1 nM E2 estradiolMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.0280nMAssay Description:Apparent binding affinity against estradiol-stimulated T-47D cell proliferationMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.0420nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 3.3%ethanolMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.0470nMAssay Description:Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol)More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.0690nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 2.5%DMFMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.0760nMAssay Description:Apparent inhibition constant for estrogen receptor in Human Breast cancer cytosol in 2.5%DMFMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.0900nMAssay Description:Apparent binding affinity against estradiol-stimulated ZR-75-1-cell proliferationMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.113nMAssay Description:Apparent inhibition constant for estrogen receptor in Human Breast cancer cytosol in 2.5%DMFMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 3.3%ethanolMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.126nMAssay Description:Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol)More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.128nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 3.3%ethanolMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.138nMAssay Description:Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol)More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.181nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 2.5%DMFMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.249nMAssay Description:Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol)More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.346nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 3.3%ethanolMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.525nMAssay Description:Apparent binding affinity against estradiol-stimulated T-47D cell proliferationMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.668nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 2.5%DMFMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 0.755nMAssay Description:Apparent inhibition constant for estrogen receptor in Human Breast cancer cytosol in 2.5%DMFMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Apparent inhibition constant for estrogen receptor in Human Breast cancer cytosol in 2.5%DMFMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 2.5%DMFMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 3.3%ethanolMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol)More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 3.3%ethanolMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Apparent binding affinity against estradiol-stimulated T-47D cell proliferationMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol)More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol)More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 7.60nMAssay Description:Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol)More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 3.3%ethanolMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol)More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: 34nMAssay Description:Apparent inhibition constant for estrogen receptor in Human uterine cytosol in 3.3%ethanolMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataKi: >270nMAssay Description:Inhibition of estradiol binding to estrogen receptor in Human Breast cancer cytosol (3.3% ethanol)More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataIC50: 0.140nMAssay Description:Inhibition of estradiol-stimulated T-47D cell proliferation.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataIC50: 0.140nMAssay Description:Inhibition of estradiol-stimulated T-47D cell proliferation.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataIC50: 0.243nMAssay Description:Inhibition of estradiol-stimulated T-47D cell proliferation.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataIC50: 0.550nMAssay Description:Inhibition of estradiol-stimulated ZR-75-1-cell proliferationMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Stimulation of alkaline phosphatase activity in human endometrial Ishikawa cells with 1 nM E2 estradiolMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Inhibition of estradiol-stimulated T-47D cell proliferation.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Inhibition of estradiol-stimulated T-47D cell proliferation.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of estradiol-stimulated ZR-75-1-cell proliferationMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Le Centre Hospitalier Universitaire De Qu£Bec
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of estradiol-stimulated T-47D cell proliferation.More data for this Ligand-Target Pair