Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50036633
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065508((R)-4-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenoxy]-4...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065516((R)-4-[2-Cyano-5-(pyridin-3-ylmethoxy)-phenoxy]-4-...)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065518(4-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenoxy]-4-o-t...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065523((R)-4-[2-Cyano-5-(isothiazol-4-ylmethoxy)-phenoxy]...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065524(5-[2-(3-Carboxy-1-o-tolyl-propoxy)-4-(thiophen-3-y...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065513(4-[2-Oxazol-2-yl-5-(thiophen-3-ylmethoxy)-phenoxy]...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065525(4-[2-(1H-Pyrazol-3-yl)-5-(thiophen-3-ylmethoxy)-ph...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065515((R)-4-[2-Cyano-5-(pyridin-4-ylmethoxy)-phenoxy]-4-...)
Affinity DataIC50:  20nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065521(4-[2-Acetyl-5-(thiophen-3-ylmethoxy)-phenoxy]-4-o-...)
Affinity DataIC50:  26nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065512(4-[2-Carbamoyl-5-(thiophen-3-ylmethoxy)-phenoxy]-4...)
Affinity DataIC50:  29nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065520(4-[2-Pyridin-2-yl-5-(thiophen-3-ylmethoxy)-phenoxy...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065522((R)-4-[5-(Benzo[1,3]dioxol-5-ylmethoxy)-2-cyano-ph...)
Affinity DataIC50:  69nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065514(5-Oxo-5-[3-(thiophen-3-ylmethoxy)-phenyl]-4-o-toly...)
Affinity DataIC50:  110nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065511((S)-4-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenoxy]-4...)
Affinity DataIC50:  113nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065510(2-(3-Carboxy-1-o-tolyl-propoxy)-4-(thiophen-3-ylme...)
Affinity DataIC50:  207nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065507(4-[3-(Thiophen-3-ylmethoxy)-phenoxy]-4-o-tolyl-but...)
Affinity DataIC50:  871nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065517(5-(2,4-Bis-benzyloxy-phenyl)-1H-pyrazole-3-carboxy...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065524(5-[2-(3-Carboxy-1-o-tolyl-propoxy)-4-(thiophen-3-y...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065518(4-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenoxy]-4-o-t...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065516((R)-4-[2-Cyano-5-(pyridin-3-ylmethoxy)-phenoxy]-4-...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065521(4-[2-Acetyl-5-(thiophen-3-ylmethoxy)-phenoxy]-4-o-...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065509(4-[2-(1H-Imidazol-2-yl)-5-(thiophen-3-ylmethoxy)-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065508((R)-4-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenoxy]-4...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065512(4-[2-Carbamoyl-5-(thiophen-3-ylmethoxy)-phenoxy]-4...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065523((R)-4-[2-Cyano-5-(isothiazol-4-ylmethoxy)-phenoxy]...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065525(4-[2-(1H-Pyrazol-3-yl)-5-(thiophen-3-ylmethoxy)-ph...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065522((R)-4-[5-(Benzo[1,3]dioxol-5-ylmethoxy)-2-cyano-ph...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065511((S)-4-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenoxy]-4...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065520(4-[2-Pyridin-2-yl-5-(thiophen-3-ylmethoxy)-phenoxy...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
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Curated by ChEMBL
LigandPNGBDBM50065510(2-(3-Carboxy-1-o-tolyl-propoxy)-4-(thiophen-3-ylme...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065513(4-[2-Oxazol-2-yl-5-(thiophen-3-ylmethoxy)-phenoxy]...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065515((R)-4-[2-Cyano-5-(pyridin-4-ylmethoxy)-phenoxy]-4-...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065507(4-[3-(Thiophen-3-ylmethoxy)-phenoxy]-4-o-tolyl-but...)
Affinity DataIC50: >3.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065514(5-Oxo-5-[3-(thiophen-3-ylmethoxy)-phenyl]-4-o-toly...)
Affinity DataIC50: >3.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)
Affinity DataIC50: >3.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065517(5-(2,4-Bis-benzyloxy-phenyl)-1H-pyrazole-3-carboxy...)
Affinity DataIC50: >3.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065509(4-[2-(1H-Imidazol-2-yl)-5-(thiophen-3-ylmethoxy)-p...)
Affinity DataIC50:  1.63E+5nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed