Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50008180
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071302(6-(2-Benzyl-thiazol-4-yl)-5-methoxy-pyridine-2-car...)
Affinity DataIC50:  860nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071304(5-Methoxy-6-(2-phenethyl-thiazol-4-yl)-pyridine-2-...)
Affinity DataIC50:  980nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071317(6-(2-Heptyl-thiazol-4-yl)-4,5-dimethoxy-pyridine-2...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071312(6-[2-(6-Hydroxy-heptyl)-thiazol-4-yl]-4,5-dimethox...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071306(5-Methoxy-6-(2-phenyl-thiazol-4-yl)-pyridine-2-car...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071316(4,5-Dimethoxy-6-(2-methyl-thiazol-4-yl)-pyridine-2...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071315(5-Methoxy-6-(2-methyl-thiazol-4-yl)-pyridine-2-car...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071309(5-Methoxy-6-(2-naphthalen-2-yl-thiazol-4-yl)-pyrid...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071303(6-(1H-Imidazol-4-yl)-5-methoxy-pyridine-2-carboxyl...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071311(4,5-Dimethoxy-6-(2-methylamino-thiazol-4-yl)-pyrid...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071308(4,5-Dimethoxy-6-thiazol-4-yl-pyridine-2-carboxylic...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071310(6-(2-Biphenyl-4-yl-thiazol-4-yl)-5-methoxy-pyridin...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071313(6-(2-Methyl-thiazol-4-yl)-pyridine-2-carboxylic ac...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071305(5-Methoxy-6-thiazol-2-yl-pyridine-2-carboxylic aci...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071314(6-Furan-3-yl-4,5-dimethoxy-pyridine-2-carboxylic a...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071301(4,5-Dimethoxy-6-(1-methyl-1H-pyrrol-2-yl)-pyridine...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50071307(4,5-Dimethoxy-6-thiophen-3-yl-pyridine-2-carboxyli...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed