Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 2001
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350315(US10208064, Example 30)
Affinity DataIC50:  6nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350299(US10208064, Example 18)
Affinity DataIC50:  7nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350282(US10208064, Example 2)
Affinity DataIC50:  9nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350300(US10208064, Example 19)
Affinity DataIC50:  10nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350301(US10208064, Example 20)
Affinity DataIC50:  11nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350289(US10208064, Example 8)
Affinity DataIC50:  13nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350296(US10208064, Example 15)
Affinity DataIC50:  14nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350305(US10208064, Example 24)
Affinity DataIC50:  16nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350304(US10208064, Example 23)
Affinity DataIC50:  17nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350312(8-(2-hydroxy-1-(tetrazolo[1,5-a]quinolin-7-yl)ethy...)
Affinity DataIC50:  18nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350302(US10208064, Example 21)
Affinity DataIC50:  19nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350290(US10208064, Example 9)
Affinity DataIC50:  19nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350298(US10208064, Example 17)
Affinity DataIC50:  20nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350294(US10208064, Example 13)
Affinity DataIC50:  23nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350309(8-(2-hydroxy-2-((R)-5-methyl-5H-tetrazolo[5,1-^...)
Affinity DataIC50:  27nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350311(8-((S)-2-hydroxy-2-((R)-5-methyl-5H-tetrazolo[5,1-...)
Affinity DataIC50:  29nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350281(US10208064, Example 1)
Affinity DataIC50:  31nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350297(US10208064, Example 16)
Affinity DataIC50:  32nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350287((R)-8-(2-(4,5-dihydrotetrazolo[1,5-a]quinolin-7-yl...)
Affinity DataIC50:  34nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350283(US10208064, Example 3)
Affinity DataIC50:  35nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350310(8-((R)-2-hydroxy-2-((R)-5-methyl-5H-tetrazolo[5,1-...)
Affinity DataIC50:  36nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350288((S)-8-(2-(4,5-dihydrotetrazolo[1,5-a]quinolin-7-yl...)
Affinity DataIC50:  38nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350286(US10208064, Example 6)
Affinity DataIC50:  40nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350284(US10208064, Example 4)
Affinity DataIC50:  43nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350313((S)-8-(2-hydroxy-1-(tetrazolo[1,5-a]quinolin-7-yl)...)
Affinity DataIC50:  44nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350291(US10208064, Example 10)
Affinity DataIC50:  46nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350292(US10208064, Example 11)
Affinity DataIC50:  47nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350307(US10208064, Example 26)
Affinity DataIC50:  82nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350308(8-(2-hydroxy-2-((S)-5-methyl-5H-tetrazolo[5,1-^...)
Affinity DataIC50:  87nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350285(US10208064, Example 5)
Affinity DataIC50:  111nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350306(US10208064, Example 25)
Affinity DataIC50:  128nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350303(US10208064, Example 22)
Affinity DataIC50:  185nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350293(US10208064, Example 12)
Affinity DataIC50:  188nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350316(US10208064, Example 31)
Affinity DataIC50:  239nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350295(US10208064, Example 14)
Affinity DataIC50:  284nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Wuxi Apptec (Shanghai)

US Patent
LigandPNGBDBM350314(US10208064, Example 29)
Affinity DataIC50:  421nMAssay Description:A Thallium Flux Assay was performed on the compounds of the Examples. This assay has been described previously; see, e.g., PCT Published Application ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent